SCHEMBL3398779

SCHEMBL3398779

CCN(CC)CCN(C)C(=O)c1sc(-c2cc(C(F)(F)F)cc(C(F)(F)F)c2)nc1C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 5/20 0.48
ALDH1A1 P00352 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
NPC1 O15118 2/20 0.45
GAA P10253 1/20 0.45
HDAC4 P56524 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
HTR2C P28335 2/20 0.41
MAPT P10636 5/20 0.41
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
TRPM8 Q7Z2W7 1/20 0.39
KDM4E B2RXH2 1/20 0.39
HSP90AA1 P07900 1/20 0.39
CRHBP P24387 1/20 0.39
CRHR2 Q13324 1/20 0.39
NR1H4 Q96RI1 1/20 0.38
CTSK P43235 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3405267 0.90 ALDH1A1 (0.63) PPARAALDH1A1SMN1; SMN2NPC1GAA
SCHEMBL3399563 0.85 HTR2C (0.43) PPARAALDH1A1SMN1; SMN2NPC1GAA
SCHEMBL3405714 0.85 HTR2C (0.45) PPARAALDH1A1SMN1; SMN2NPC1GAA
SCHEMBL3404493 0.83 KMT2A (0.44) PPARAALDH1A1SMN1; SMN2NPC1GAA
SCHEMBL13309741 0.83 RAB9A (0.56) PPARAALDH1A1SMN1; SMN2NPC1GAA
SCHEMBL3403383 0.82 PPARA (0.44) PPARAALDH1A1SMN1; SMN2NPC1GAA
SCHEMBL3405487 0.82 HTR2C (0.44) PPARAALDH1A1SMN1; SMN2NPC1GAA
SCHEMBL3404554 0.81 HTR2C (0.44) PPARAALDH1A1SMN1; SMN2NPC1GAA
SCHEMBL3400845 0.81 PPARA (0.51) PPARAALDH1A1SMN1; SMN2NPC1GAA
SCHEMBL3404118 0.80 PPARA (0.57) PPARAALDH1A1NPC1GAAHDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
WO-2006089076-A9 THIAZOLE AMIDES, IMIDAZOLE AMIDES AND RELATED ANALOGUES NEUROGEN CORP (US) 2007-04-26 WO disclosed