SCHEMBL3400514

SCHEMBL3400514

CCCCN1CCCN(C(=O)c2sc(-c3ccc4ccccc4c3)nc2C)CC1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 7/20 0.48
CNR1 P21554 1/20 0.48
THRA P10827 2/20 0.45
THRB P10828 2/20 0.45
HRH3 Q9Y5N1 1/20 0.43
CES2 O00748 1/20 0.41
GRIN2B Q13224 2/20 0.41
PARP1 P09874 3/20 0.40
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3402959 0.91 HRH3 (0.46) HTR2CCNR1THRATHRBHRH3
SCHEMBL3401176 0.89 CNR1 (0.60) HTR2CCNR1HRH3CES2PARP1
SCHEMBL3402609 0.89 THRA (0.47) HTR2CCNR1THRATHRBHRH3
SCHEMBL3405569 0.88 CNR1 (0.48) HTR2CCNR1THRATHRBHRH3
SCHEMBL3402322 0.87 CNR1 (0.46) HTR2CCNR1THRATHRBHRH3
SCHEMBL3403844 0.87 CNR1 (0.51) HTR2CCNR1THRATHRBHRH3
SCHEMBL3405885 0.87 THRA (0.45) HTR2CCNR1THRATHRBHRH3
SCHEMBL3400494 0.87 THRA (0.45) HTR2CCNR1THRATHRBHRH3
SCHEMBL3404391 0.86 CNR1 (0.46) HTR2CCNR1THRATHRBHRH3
SCHEMBL3403653 0.86 THRA (0.45) HTR2CCNR1THRATHRBHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
WO-2006089076-A9 THIAZOLE AMIDES, IMIDAZOLE AMIDES AND RELATED ANALOGUES NEUROGEN CORP (US) 2007-04-26 WO disclosed