SCHEMBL3400535

SCHEMBL3400535

C=CCC(N)(CCC(N)[C@@](C)(I)c1ccc(Br)cc1)c1ccccc1

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.35
KIF11 P52732 5/20 0.33
ALDH1A1 P00352 1/20 0.31
TSHR P16473 1/20 0.31
ATM Q13315 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3194342 0.78 HTR2A (0.33) HTTKIF11ALDH1A1TSHR
SCHEMBL30434709 0.70 HTT (0.46) HTTKIF11ALDH1A1TSHRATM
SCHEMBL9962944 0.69 LMNA (0.36) HTTALDH1A1ATM
SCHEMBL830678 0.69 PYCR1 (0.37) HTTALDH1A1TSHRATM
SCHEMBL2688608 0.68 HTT (0.53) HTTKIF11ALDH1A1TSHRATM
Hydrochloric Acid SCHEMBL11764056 0.67 HTT (0.52) HTTKIF11ALDH1A1TSHRATM
SCHEMBL7131764 0.66 HTT (0.45) HTTALDH1A1TSHRATM
SCHEMBL8508636 0.65 HTT (0.44) HTTKIF11ALDH1A1TSHRATM
SCHEMBL9593286 0.64 HTT (0.49) HTTKIF11ALDH1A1TSHRATM
SCHEMBL30434781 0.64 PYCR1 (0.36) HTTALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2252598-A2 1,3-OXAZEPAN-2-ONE AND 1,3-DIAZEPAN-2-ONE INHIBITORS OF 11BETA-HYDROXYSTEROID DEHYDROGENASE 1 Vitae Pharmaceuticals, Inc. (US) 2010-11-24 EP disclosed
WO-2009102428-A2 1,3-OXAZEPAN-2-ONE AND 1,3-DIAZEPAN-2-ONE INHIBITORS OF 11β -HYDROXYSTEROID DEHYDROGENASE 1 VITAE PHARMACEUTICALS, INC. (US) 2009-08-20 WO disclosed