SCHEMBL3401005

SCHEMBL3401005

CC(C)(C)CNC(=O)c1cnc2ccccc2c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 3/20 0.56
MGAM O43451 1/20 0.55
HDAC3 O15379 2/20 0.54
HDAC1 Q13547 2/20 0.54
HDAC2 Q92769 1/20 0.54
BCAT1 P54687 1/20 0.51
TRPV1 Q8NER1 1/20 0.51
PPARD Q03181 1/20 0.51
PREP P48147 1/20 0.50
MEN1 O00255 1/20 0.48
MAPT P10636 1/20 0.48
KMT2A Q03164 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CFTR P13569 1/20 0.48
KDR P35968 1/20 0.48
KDM4E B2RXH2 1/20 0.47
NPC1 O15118 1/20 0.47
MITF O75030 1/20 0.47
XBP1 P17861 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13113540 0.82 MGAM (0.56) HPGDSMGAMHDAC3HDAC1HDAC2
SCHEMBL7209315 0.81 MGAM (0.59) HPGDSMGAMHDAC3HDAC1HDAC2
SCHEMBL20812002 0.81 HPGDS (0.65) HPGDSMGAMHDAC3HDAC1HDAC2
SCHEMBL5309154 0.80 MGAM (0.62) HPGDSMGAMHDAC3HDAC1HDAC2
SCHEMBL10242977 0.80 HDAC3 (0.61) HPGDSMGAMHDAC3HDAC1HDAC2
SCHEMBL6237473 0.79 MGAM (0.65) HPGDSMGAMHDAC3HDAC1HDAC2
SCHEMBL22389 0.79 PLK1 (0.65) HPGDSMGAMHDAC3HDAC1HDAC2
SCHEMBL24392693 0.79 HPGDS (0.70) HPGDSMGAMHDAC3HDAC1HDAC2
SCHEMBL30858823 0.79 HDAC3 (0.61) HPGDSMGAMHDAC3HDAC1HDAC2
SCHEMBL29222038 0.79 HDAC3 (0.61) HPGDSMGAMHDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2252611-A1 (DIHYDRO)PYRROLO[2,1-A]ISOQUINOLINES N.V. Organon (NL) 2010-11-24 EP disclosed
WO-2009098283-A1 (DIHYDRO)PYRROLO[2,1-A]ISOQUINOLINES N.V. ORGANON (NL) 2009-08-13 WO disclosed