SCHEMBL3401280

SCHEMBL3401280

Cc1nc(-c2ccc(F)cc2F)sc1C(=O)NCCCN1CCCC1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.48
GAA P10253 1/20 0.47
SMYD2 Q9NRG4 5/20 0.46
MKNK2 Q9HBH9 3/20 0.45
MAPT P10636 2/20 0.45
ULK1 O75385 1/20 0.44
STAT3 P40763 2/20 0.43
KMT2A Q03164 1/20 0.43
NAMPT P43490 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3404848 0.97 RAB9A (0.45) RAB9AGAASMYD2MKNK2MAPT
SCHEMBL3396887 0.94 RAB9A (0.48) RAB9AGAASMYD2MKNK2MAPT
SCHEMBL3405409 0.94 SCN9A (0.47) RAB9ASTAT3
SCHEMBL3401224 0.93 SCN9A (0.49) RAB9AGAASTAT3
SCHEMBL3401313 0.88 SCN9A (0.47) STAT3
SCHEMBL3400482 0.88 DRD2 (0.46) GAASMYD2MAPTKMT2A
SCHEMBL3405360 0.87 SCN9A (0.49) GAASTAT3
SCHEMBL3402323 0.85 DPP4 (0.49) GAA
SCHEMBL3402585 0.84 DRD2 (0.47) SMYD2MKNK2
SCHEMBL3402094 0.84 DPP4 (0.50) GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
WO-2006089076-A9 THIAZOLE AMIDES, IMIDAZOLE AMIDES AND RELATED ANALOGUES NEUROGEN CORP (US) 2007-04-26 WO disclosed