SCHEMBL3405409

SCHEMBL3405409

Cc1nc(-c2ccc(F)cc2F)sc1C(=O)NCCN1CCCC1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 4/20 0.47
TSHR P16473 2/20 0.45
SRC P12931 1/20 0.45
CACNA1G O43497 3/20 0.43
NPSR1 Q6W5P4 1/20 0.43
RAB9A P51151 1/20 0.43
CHRM4 P08173 1/20 0.42
PDGFRB P09619 1/20 0.42
FGFR1 P11362 1/20 0.42
KDR P35968 1/20 0.42
TLK2 Q86UE8 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C19 P33261 1/20 0.42
STAT3 P40763 1/20 0.42
PARP1 P09874 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3401224 0.99 SCN9A (0.49) SCN9ATSHRSRCCACNA1GNPSR1
SCHEMBL3401280 0.94 RAB9A (0.48) RAB9ASTAT3
SCHEMBL3401313 0.94 SCN9A (0.47) SCN9ATSHRSRCCACNA1GNPSR1
SCHEMBL3404848 0.93 RAB9A (0.45) SCN9ARAB9ASTAT3
SCHEMBL3405360 0.93 SCN9A (0.49) SCN9ATSHRSRCCACNA1GNPSR1
SCHEMBL3402323 0.90 DPP4 (0.49) SCN9ACACNA1GNPSR1CHRM4
SCHEMBL3402094 0.89 DPP4 (0.50) SCN9ACACNA1GCHRM4
SCHEMBL3396887 0.88 RAB9A (0.48) RAB9APDGFRBKDRSTAT3
SCHEMBL3403561 0.84 WNT1 (0.52) SCN9ATSHRNPSR1CHRM4PARP1
SCHEMBL13309881 0.84 ACKR3 (0.54) CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
WO-2006089076-A9 THIAZOLE AMIDES, IMIDAZOLE AMIDES AND RELATED ANALOGUES NEUROGEN CORP (US) 2007-04-26 WO disclosed