SCHEMBL3401416

SCHEMBL3401416

Cc1nc(-c2ccccc2Cl)sc1C(=O)NCCN1CCCCC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.53
ALDH1A1 P00352 2/20 0.53
MAPT P10636 1/20 0.53
RAB9A P51151 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
PDE2A O00408 2/20 0.52
PDE10A Q9Y233 1/20 0.52
PPARD Q03181 1/20 0.50
PPARA Q07869 1/20 0.50
CHRM4 P08173 2/20 0.49
HTR2C P28335 1/20 0.47
PARP1 P09874 1/20 0.46
LMNA P02545 1/20 0.45
NPSR1 Q6W5P4 2/20 0.45
SMYD2 Q9NRG4 1/20 0.45
CACNA1G O43497 2/20 0.45
HPGD P15428 1/20 0.45
APP P05067 1/20 0.44
KDM4E B2RXH2 1/20 0.43
HSD17B10 Q99714 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3402762 0.99 NPC1 (0.53) NPC1ALDH1A1MAPTRAB9ASMN1; SMN2
SCHEMBL3402982 0.93 SMYD2 (0.53) NPC1ALDH1A1MAPTRAB9ASMN1; SMN2
SCHEMBL3405595 0.92 PDE2A (0.47) NPC1ALDH1A1MAPTRAB9ASMN1; SMN2
SCHEMBL3403787 0.92 SMYD2 (0.50) NPC1ALDH1A1MAPTRAB9ASMN1; SMN2
SCHEMBL3401250 0.91 PDE2A (0.47) NPC1ALDH1A1MAPTRAB9ASMN1; SMN2
SCHEMBL3405826 0.88 DPP4 (0.49) ALDH1A1PDE2APDE10ACHRM4NPSR1
SCHEMBL3400943 0.88 DPP4 (0.56) ALDH1A1MAPTPPARACHRM4CACNA1G
SCHEMBL3398247 0.87 ALDH1A1 (0.48) ALDH1A1SMN1; SMN2PDE2APDE10ACHRM4
SCHEMBL3401355 0.87 DPP4 (0.54) ALDH1A1MAPTSMN1; SMN2PDE2APDE10A
SCHEMBL3401847 0.86 HTR2C (0.45) NPC1SMN1; SMN2PDE2APDE10ACHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
WO-2006089076-A9 THIAZOLE AMIDES, IMIDAZOLE AMIDES AND RELATED ANALOGUES NEUROGEN CORP (US) 2007-04-26 WO disclosed