SCHEMBL3405595

SCHEMBL3405595

Cc1nc(-c2cccc(Cl)c2Cl)sc1C(=O)NCCN1CCCCC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 1/20 0.47
PDE10A Q9Y233 1/20 0.47
HTR2C P28335 7/20 0.45
CHRM4 P08173 1/20 0.45
PPARD Q03181 1/20 0.45
PPARA Q07869 1/20 0.45
HTR2A P28223 4/20 0.45
SLC6A4 P31645 4/20 0.45
LMNA P02545 1/20 0.44
PANK3 Q9H999 1/20 0.44
ALDH1A1 P00352 3/20 0.44
NPC1 O15118 1/20 0.44
MAPT P10636 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
TSHR P16473 1/20 0.43
DRD2 P14416 2/20 0.43
PARP1 P09874 1/20 0.43
HTR1A P08908 1/20 0.43
DRD4 P21917 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3401250 0.99 PDE2A (0.47) PDE2APDE10AHTR2CCHRM4PPARD
SCHEMBL3396859 0.92 DRD2 (0.51) HTR2CHTR2ASLC6A4DRD2HTR1A
SCHEMBL3401416 0.92 NPC1 (0.53) PDE2APDE10AHTR2CCHRM4PPARD
SCHEMBL3402762 0.91 NPC1 (0.53) PDE2APDE10AHTR2CCHRM4PPARD
SCHEMBL3402982 0.85 SMYD2 (0.53) PDE2APDE10ACHRM4PPARDPPARA
SCHEMBL3400943 0.84 DPP4 (0.56) CHRM4PPARAALDH1A1MAPTDRD2
SCHEMBL3405826 0.84 DPP4 (0.49) PDE2APDE10ACHRM4ALDH1A1DRD2
SCHEMBL3403787 0.84 SMYD2 (0.50) PDE2APDE10ACHRM4PPARDPPARA
SCHEMBL3398247 0.83 ALDH1A1 (0.48) PDE2APDE10ACHRM4ALDH1A1SMN1; SMN2
SCHEMBL3401355 0.83 DPP4 (0.54) PDE2APDE10ACHRM4PPARDPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
US-7728009-B1 Thiazole amides, imidazole amides and related analogues NEUROGEN CORPORATION (US) 2010-06-01 US disclosed
WO-2006089076-A9 THIAZOLE AMIDES, IMIDAZOLE AMIDES AND RELATED ANALOGUES NEUROGEN CORP (US) 2007-04-26 WO disclosed