SCHEMBL3401547

SCHEMBL3401547

CCOC(=O)c1c(Cl)c(CC(=O)c2ccccc2)c(C)[nH]c1=O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.53
HPGD P15428 1/20 0.53
NPC1 O15118 8/20 0.50
RAB9A P51151 7/20 0.50
CASP3 P42574 1/20 0.50
SENP8 Q96LD8 1/20 0.50
SENP7 Q9BQF6 1/20 0.50
SENP6 Q9GZR1 1/20 0.50
MAPT P10636 6/20 0.47
SMN1; SMN2 Q16637 4/20 0.47
CSF1R P07333 1/20 0.46
MAP3K5 Q99683 1/20 0.43
LMNA P02545 3/20 0.43
KMT2A Q03164 4/20 0.43
TDP1 Q9NUW8 3/20 0.43
MEN1 O00255 3/20 0.43
POLB P06746 1/20 0.43
ALDH1A1 P00352 2/20 0.42
PDE3B Q13370 1/20 0.42
PDE3A Q14432 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7008205 0.79 CYP1A2 (0.54) KDM4EHPGDNPC1MAPTSMN1; SMN2
SCHEMBL26664855 0.73 HPGD (0.51) KDM4EHPGDNPC1MAPTSMN1; SMN2
SCHEMBL1061379 0.72 KDM4E (0.64) KDM4ERAB9AMAPTSMN1; SMN2CSF1R
SCHEMBL16972721 0.68 TP53 (0.56) KDM4EHPGDNPC1RAB9AMAPT
SCHEMBL4696686 0.68 CSF1R (0.61) KDM4EHPGDMAPTSMN1; SMN2CSF1R
SCHEMBL17952494 0.68 ALDH1A1 (0.62) KDM4EHPGDNPC1RAB9AMAPT
SCHEMBL1156774 0.68 MAPT (0.54) KDM4EHPGDNPC1RAB9ACASP3
SCHEMBL5188877 0.68 CYP1A2 (0.60) KDM4EHPGDNPC1MAPTSMN1; SMN2
Ethyl Benzoate SCHEMBL11244230 0.68 LMNA (0.68) NPC1RAB9AMAPTSMN1; SMN2LMNA
SCHEMBL11277059 0.67 MAP3K5 (0.54) KDM4EHPGDNPC1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2247588-A2 FUSED HETEROCYCLIC DERIVATIVE AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2010-11-10 EP disclosed
WO-2009107850-A2 FUSED HETEROCYCLIC DERIVATIVE AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-09-03 WO disclosed