SCHEMBL3401694

SCHEMBL3401694

COc1ccc(NNc2cccc(OCCN3CCOCC3)c2)cc1OCCN1CCOCC1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.54
TSHR P16473 3/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
NPSR1 Q6W5P4 1/20 0.54
HTR2C P28335 2/20 0.52
HTR2B P41595 2/20 0.52
SRC P12931 1/20 0.52
KDR P35968 1/20 0.52
CYP2D6 P10635 1/20 0.51
EPHX2 P34913 6/20 0.50
KDM4E B2RXH2 2/20 0.49
HTT P42858 1/20 0.49
POLB P06746 1/20 0.48
TP53 P04637 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3401693 0.81 HTR2C (0.55) ALDH1A1TSHRSMN1; SMN2NPSR1HTR2C
SCHEMBL14621966 0.80 EPHX2 (0.59) ALDH1A1TSHRSMN1; SMN2NPSR1EPHX2
SCHEMBL14578174 0.80 EPHX2 (0.61) ALDH1A1TSHRSMN1; SMN2NPSR1SRC
SCHEMBL13791083 0.79 SYK (0.59) ALDH1A1TSHRSMN1; SMN2NPSR1HTR2C
SCHEMBL3548030 0.78 NPC1 (0.52) ALDH1A1TSHRSMN1; SMN2NPSR1SRC
SCHEMBL5319656 0.78 KDM4E (0.70) ALDH1A1TSHRSMN1; SMN2CYP2D6KDM4E
SCHEMBL12837450 0.78 ALDH1A1 (0.60) ALDH1A1TSHRSMN1; SMN2NPSR1EPHX2
Ammonia Solution, Strong SCHEMBL4267670 0.77 KDM4E (0.68) ALDH1A1TSHRSMN1; SMN2CYP2D6KDM4E
SCHEMBL12764910 0.77 EPHX2 (0.63) ALDH1A1TSHRSMN1; SMN2NPSR1EPHX2
SCHEMBL7010009 0.77 HTR2C (0.49) TSHRHTR2CHTR2BKDRCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2247591-A1 PYRROLO [2, 3-D]PYRIDINES AND USE THEREOF AS TYROSINE KINASE INHIBITORS Novartis AG (CH) 2010-11-10 EP disclosed
WO-2009098236-A1 PYRROLO [2, 3-D] PYRIDINES AND USE THEREOF AS TYROSINE KINASE INHIBITORS NOVARTIS AG (CH) 2009-08-13 WO disclosed