SCHEMBL3401971

SCHEMBL3401971

CC(C)(C(=O)N1CCOCC1)c1ccc(Br)cc1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.55
AKR1C3 P42330 1/20 0.51
MGLL Q99685 2/20 0.50
PHGDH O43175 1/20 0.50
POLB P06746 1/20 0.49
RAB9A P51151 5/20 0.48
KMT2A Q03164 3/20 0.48
MEN1 O00255 2/20 0.48
NPC1 O15118 4/20 0.46
HSD17B10 Q99714 2/20 0.46
ALDH1A1 P00352 2/20 0.46
HPGD P15428 2/20 0.46
MAPT P10636 2/20 0.45
GAA P10253 1/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
NR1I2 O75469 1/20 0.43
KCNH2 Q12809 1/20 0.43
GRM2 Q14416 1/20 0.43
ALOX15 P16050 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19070596 0.84 SMN1; SMN2 (0.77) SMN1; SMN2AKR1C3PHGDHRAB9AHPGD
SCHEMBL15023275 0.82 SMN1; SMN2 (0.56) SMN1; SMN2POLBRAB9AKMT2AMEN1
SCHEMBL16464172 0.81 SMN1; SMN2 (0.55) SMN1; SMN2MGLLPOLBRAB9AKMT2A
SCHEMBL16625322 0.76 HSD11B1 (0.38) POLBRAB9AKMT2AMEN1NPC1
SCHEMBL17796641 0.76 AKR1C3 (0.52) SMN1; SMN2AKR1C3PHGDHPOLBRAB9A
SCHEMBL28941604 0.74 SMN1; SMN2 (0.56) SMN1; SMN2MGLLRAB9AKMT2AMEN1
SCHEMBL28770085 0.74 SMN1; SMN2 (0.47) SMN1; SMN2RAB9AKMT2AMEN1NPC1
SCHEMBL12477371 0.72 ALDH1A1 (0.55) SMN1; SMN2AKR1C3RAB9AKMT2AMEN1
SCHEMBL12477377 0.72 ALDH1A1 (0.55) SMN1; SMN2AKR1C3RAB9AKMT2AMEN1
SCHEMBL18644455 0.72 RAB9A (0.58) SMN1; SMN2AKR1C3POLBRAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2247591-A1 PYRROLO [2, 3-D]PYRIDINES AND USE THEREOF AS TYROSINE KINASE INHIBITORS Novartis AG (CH) 2010-11-10 EP disclosed
WO-2009098236-A1 PYRROLO [2, 3-D] PYRIDINES AND USE THEREOF AS TYROSINE KINASE INHIBITORS NOVARTIS AG (CH) 2009-08-13 WO disclosed