SCHEMBL3403177

SCHEMBL3403177

c1ccc2[nH]c(Cc3ccc4c(n3)C(NCc3ccc(-n5ccnc5)cc3)CCC4)nc2c1

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 15/20 0.41
TAOK1 Q7L7X3 1/20 0.38
TAOK3 Q9H2K8 1/20 0.38
CHRM2 P08172 1/20 0.36
CYP2D6 P10635 1/20 0.36
DRD2 P14416 1/20 0.36
OPRM1 P35372 1/20 0.36
KCNH2 Q12809 1/20 0.36
SLC40A1 Q9NP59 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4881182 0.77 CXCR4 (0.46) CXCR4
SCHEMBL2509452 0.73 CXCR4 (0.73) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL4760826 0.71 CXCR4 (0.49) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL31257251 0.70 SLC40A1 (0.59) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL3370850 0.70 SLC40A1 (0.59) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL4760828 0.70 SLC40A1 (0.59) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL7104696 0.68 CXCR4 (0.61) CXCR4
SCHEMBL31059309 0.68 CXCR4 (0.61) CXCR4
SCHEMBL4069397 0.68 CXCR4 (0.76) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL7407358 0.68 CBFB (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1752455-B1 Chemokine receptor binding heterocyclic compounds ANORMED INC (CA) 2010-11-10 EP claimed