SCHEMBL3405757

SCHEMBL3405757

CCC(NC(=O)c1cnc(-c2cc(Br)ccn2)nc1O)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.48
KDM4E B2RXH2 1/20 0.48
LMNA P02545 1/20 0.48
HPGD P15428 1/20 0.48
TSHR P16473 1/20 0.48
HSD17B10 Q99714 1/20 0.48
TACR3 P29371 8/20 0.48
TACR2 P21452 4/20 0.48
PDE2A O00408 1/20 0.43
KCNK3 O14649 4/20 0.42
ROCK1 Q13464 2/20 0.42
MAPT P10636 1/20 0.41
HTT P42858 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
KCNA5 P22460 2/20 0.41
PPARG P37231 1/20 0.41
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3435595 0.89 KDM4E (0.49) ALDH1A1KDM4ELMNAHPGDTSHR
SCHEMBL16005739 0.79 ALDH1A1 (0.49) ALDH1A1KDM4ELMNAHPGDTSHR
SCHEMBL4520187 0.79 ALDH1A1 (0.49) ALDH1A1KDM4ELMNAHPGDTSHR
SCHEMBL4527992 0.79 ALDH1A1 (0.49) ALDH1A1KDM4ELMNAHPGDTSHR
SCHEMBL3405746 0.77 EGLN1 (0.52) TACR3PDE2A
SCHEMBL3434892 0.76 TSHR (0.50) ALDH1A1KDM4ELMNAHPGDTSHR
SCHEMBL4527612 0.76 KDM4E (0.45) ALDH1A1KDM4EHPGDTSHRHSD17B10
SCHEMBL3435598 0.72 EGLN1 (0.50) ALDH1A1KDM4ELMNAHPGDTSHR
SCHEMBL3410929 0.72 EGLN1 (0.50) ALDH1A1KDM4ELMNAHPGDTSHR
SCHEMBL14822498 0.70 HPGDS (0.42) ALDH1A1KDM4ELMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2257539-A1 SUBSTITUTED 4-HYDROXYPYRIMIDINE-5-CARBOXAMIDES Merck Sharp & Dohme Corp. (US) 2010-12-08 EP disclosed
WO-2009117269-A1 SUBSTITUTED 4-HYDROXYPYRIMIDINE-5-CARBOXAMIDES MERCK & CO., INC. (US) 2009-09-24 WO disclosed