SCHEMBL3406569

SCHEMBL3406569

CC(C)n1c(Cn2ccnc2-c2ncccc2F)nc2cccnc21

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 2/20 0.35
NPC1 O15118 1/20 0.35
PKM P14618 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ENPP2 Q13822 6/20 0.34
TP53 P04637 5/20 0.34
MAPT P10636 1/20 0.34
LMNA P02545 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
PDE2A O00408 1/20 0.33
POLB P06746 1/20 0.33
PABPC1 P11940 1/20 0.33
ADORA2A P29274 1/20 0.32
ADORA1 P30542 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3059903 0.87 PDE10A (0.35) PDE10AENPP2TP53MAPTLMNA
SCHEMBL3068576 0.83 TP53 (0.38) PDE10ANPC1PKMRAB9ASMN1; SMN2
SCHEMBL3060632 0.82 TP53 (0.43) PDE10ANPC1PKMRAB9ASMN1; SMN2
SCHEMBL3070806 0.80 ENPP2 (0.36) NPC1PKMRAB9ASMN1; SMN2ENPP2
SCHEMBL3067932 0.80 TP53 (0.44) SMN1; SMN2TP53MAPTLMNAPOLB
SCHEMBL3055020 0.80 AGTR2 (0.37) PDE10ARAB9AENPP2TP53MEN1
SCHEMBL3064818 0.79 ENPP2 (0.35) NPC1PKMRAB9ASMN1; SMN2ENPP2
SCHEMBL3060545 0.74 PDE10A (0.33) PDE10AMEN1KMT2AADORA2AADORA1
SCHEMBL13089466 0.74 GRM2 (0.34) PDE10ATP53
SCHEMBL3062897 0.73 PKM (0.36) PDE10APKMLMNAADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1368342-B3 BENZIMIDAZOLE AND PYRIDYLIMIDAZOLE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS NEUROGEN CORP (US) 2010-12-01 EP disclosed