SCHEMBL3407436

SCHEMBL3407436

CCOC(=O)NNc1ccc(OCc2csc(NC(C)=O)n2)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.65
SMN1; SMN2 Q16637 5/20 0.65
NPC1 O15118 4/20 0.65
LMNA P02545 5/20 0.60
HTT P42858 4/20 0.60
ALDH1A1 P00352 3/20 0.60
CASP3 P42574 1/20 0.60
SENP8 Q96LD8 1/20 0.60
SENP7 Q9BQF6 1/20 0.60
SENP6 Q9GZR1 1/20 0.60
MAPT P10636 7/20 0.51
MAPK1 P28482 4/20 0.48
KMT2A Q03164 3/20 0.48
MEN1 O00255 2/20 0.48
TP53 P04637 2/20 0.48
KDM4E B2RXH2 2/20 0.46
GAA P10253 1/20 0.45
TSHR P16473 1/20 0.44
POLB P06746 1/20 0.44
HSP90AA1 P07900 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3406120 0.85 AOC3 (0.61) RAB9ASMN1; SMN2NPC1MAPTKMT2A
SCHEMBL3403640 0.81 EGFR (0.51) RAB9ASMN1; SMN2NPC1ALDH1A1MAPT
Hydrochloric Acid SCHEMBL3402973 0.80 EGFR (0.50) RAB9ASMN1; SMN2NPC1LMNAALDH1A1
SCHEMBL6796683 0.79 NPC1 (0.77) RAB9ASMN1; SMN2NPC1LMNAHTT
SCHEMBL3405939 0.79 RAB9A (0.77) RAB9ASMN1; SMN2NPC1LMNAHTT
SCHEMBL4871628 0.79 RAB9A (1.00) RAB9ASMN1; SMN2NPC1LMNAHTT
SCHEMBL16556647 0.79 NPC1 (0.72) RAB9ASMN1; SMN2NPC1LMNAHTT
SCHEMBL3400713 0.78 AOC3 (0.55) RAB9ASMN1; SMN2NPC1LMNAHTT
SCHEMBL16242472 0.78 NPC1 (0.73) RAB9ASMN1; SMN2NPC1LMNAHTT
SCHEMBL3406292 0.77 SMN1; SMN2 (0.54) RAB9ASMN1; SMN2NPC1LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2252604-A1 THIAZOLE DERIVATIVE AND USE THEREOF AS VAP-1 INHIBITOR R-Tech Ueno, Ltd. (JP) 2010-11-24 EP claimed
WO-2009096609-A1 THIAZOLE DERIVATIVE AND USE THEREOF AS VAP-1 INHIBITOR R-TECH UENO, LTD. (JP) 2009-08-06 WO claimed
EP-2252604-A1 THIAZOLE DERIVATIVE AND USE THEREOF AS VAP-1 INHIBITOR R-Tech Ueno, Ltd. (JP) 2010-11-24 EP disclosed
WO-2009096609-A1 THIAZOLE DERIVATIVE AND USE THEREOF AS VAP-1 INHIBITOR R-TECH UENO, LTD. (JP) 2009-08-06 WO disclosed