SCHEMBL3407767

SCHEMBL3407767

Cc1c(C(COc2ccccc2)Nc2ccccc2C(=O)NCCC(=O)O)oc2ccccc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 0.45
L3MBTL1 Q9Y468 4/20 0.45
KDM4E B2RXH2 4/20 0.45
HTT P42858 2/20 0.45
MAPT P10636 2/20 0.45
TDP1 Q9NUW8 1/20 0.45
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
NPSR1 Q6W5P4 3/20 0.40
TP53 P04637 1/20 0.40
GCG P01275 1/20 0.40
PPARG P37231 1/20 0.40
GAA P10253 1/20 0.40
CA12 O43570 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
NPY1R P25929 1/20 0.39
ALDH1A1 P00352 2/20 0.39
HPGD P15428 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL719021 0.85 GCG (0.43) LMNAL3MBTL1KDM4EHTTMAPT
SCHEMBL718011 0.77 MAPT (0.42) LMNAL3MBTL1KDM4EHTTMAPT
SCHEMBL719589 0.76 NPC1 (0.48) L3MBTL1KDM4ENPC1RAB9ANPSR1
SCHEMBL718772 0.76 GCG (0.44) L3MBTL1KDM4ENPC1RAB9AGCG
SCHEMBL3400803 0.76 NPC1 (0.47) L3MBTL1KDM4ENPC1RAB9ANPSR1
SCHEMBL2669949 0.76 ADRB2 (0.44) LMNAL3MBTL1KDM4EHTTMAPT
SCHEMBL720711 0.75 CA12 (0.49) LMNAL3MBTL1KDM4EHTTMAPT
SCHEMBL721127 0.74 RAB9A (0.39) LMNAL3MBTL1KDM4EHTTMAPT
SCHEMBL719499 0.73 MAPT (0.45) LMNAL3MBTL1KDM4EMAPTNPC1
SCHEMBL716401 0.70 GCG (0.37) LMNAL3MBTL1HTTMAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2251326-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2010-11-17 EP disclosed