SCHEMBL3409641

SCHEMBL3409641

COc1cc(Nc2nccc(-c3ccc(Cl)c(C)c3)n2)ccc1-c1nc(C)c[nH]1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 7/20 0.49
PIK3CG P48736 7/20 0.49
PIK3CB P42338 6/20 0.49
EGFR P00533 3/20 0.49
JAK2 O60674 3/20 0.49
CDK2 P24941 2/20 0.49
PTK2B Q14289 1/20 0.49
RET P07949 1/20 0.43
ZAP70 P43403 5/20 0.42
CDK9 P50750 3/20 0.42
CCNT1 O60563 2/20 0.42
DYRK1A Q13627 1/20 0.42
CLK4 Q9HAZ1 1/20 0.42
PRKD3 O94806 3/20 0.42
PRKCG P05129 3/20 0.42
PRKCB P05771 3/20 0.42
LCK P06239 3/20 0.42
PRKCA P17252 3/20 0.42
PRKCH P24723 3/20 0.42
PRKCI P41743 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3407305 0.91 PIK3CA (0.61) PIK3CAPIK3CGPIK3CBEGFRJAK2
SCHEMBL3409753 0.88 PIK3CA (0.52) PIK3CAPIK3CGPIK3CBEGFRJAK2
SCHEMBL3407822 0.86 PIK3CA (0.59) PIK3CAPIK3CGPIK3CBEGFRJAK2
SCHEMBL3409953 0.86 PIK3CA (0.49) PIK3CAPIK3CGPIK3CBEGFRJAK2
SCHEMBL3413279 0.84 CDK2 (0.46) PIK3CAPIK3CGPIK3CBEGFRJAK2
SCHEMBL3408743 0.84 PRKCA (0.62) EGFRRETZAP70PRKD3PRKCG
SCHEMBL3409757 0.84 CDK9 (0.47) PIK3CAPIK3CGPIK3CBEGFRJAK2
SCHEMBL3412789 0.80 SYK (0.56) CDK2RETZAP70CDK9CCNT1
SCHEMBL3406073 0.80 PIK3CA (0.41) PIK3CAPIK3CGPIK3CBEGFRPRKCQ
SCHEMBL3412646 0.79 SYK (0.46) CDK2RETCDK9CCNT1DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2257541-A1 MODULATORS FOR AMYLOID BETA F. Hoffmann-La Roche AG (CH) 2010-12-08 EP disclosed
WO-2009103652-A1 MODULATORS FOR AMYLOID BETA F. HOFFMANN-LA ROCHE AG (CH) 2009-08-27 WO disclosed