SCHEMBL3413631

SCHEMBL3413631

COC(=O)Nc1ccc(-c2cc(CC(N)c3ccccc3)nnc2C(=O)OC)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 2/20 0.41
KDR P35968 2/20 0.41
F11 P03951 9/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
SLC1A3 P43003 2/20 0.38
SLC1A2 P43004 2/20 0.38
SLC1A1 P43005 2/20 0.38
HPGD P15428 1/20 0.38
ALDH1A1 P00352 2/20 0.37
KDM4E B2RXH2 1/20 0.37
KMT2A Q03164 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
GAA P10253 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
RORC P51449 1/20 0.36
MCL1 Q07820 1/20 0.36
KLKB1 P03952 2/20 0.35
PRSS1 P07477 1/20 0.35
PRSS2 P07478 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3413708 0.88 F11 (0.40) PDGFRBKDRF11SMN1; SMN2SLC1A3
SCHEMBL478939 0.87 F11 (0.41) PDGFRBKDRF11SMN1; SMN2SLC1A3
SCHEMBL478940 0.87 F11 (0.41) PDGFRBKDRF11SMN1; SMN2SLC1A3
SCHEMBL3413919 0.82 F11 (0.39) F11SMN1; SMN2HPGDALDH1A1KMT2A
SCHEMBL478962 0.82 F11 (0.46) PDGFRBKDRF11SMN1; SMN2NPC1
SCHEMBL478961 0.82 F11 (0.46) PDGFRBKDRF11SMN1; SMN2NPC1
SCHEMBL4707261 0.77 F11 (0.49) F11SMN1; SMN2HPGDALDH1A1KDM4E
SCHEMBL3414366 0.73 F11 (0.44) F11SMN1; SMN2HPGDKDM4ENPC1
SCHEMBL3412508 0.73 ROCK1 (0.40) F11HPGDALDH1A1KMT2ANPC1
SCHEMBL3413549 0.73 F11 (0.42) F11SMN1; SMN2HPGDNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2265601-A1 PYRIDAZINE DERIVATIVES AS FACTOR XIA INHIBITORS Bristol-Myers Squibb Company (US) 2010-12-29 EP disclosed
WO-2009114677-A1 PYRIDAZINE DERIVATIVES AS FACTOR XIA INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2009-09-17 WO disclosed