SCHEMBL3416112

SCHEMBL3416112

O=C(O)NCc1cc(Br)ccc1OCc1ccccc1.OCc1cc(Br)ccc1OCc1ccccc1

nearest known ligand 0.65

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
USP28 Q96RU2 1/20 0.65
USP25 Q9UHP3 1/20 0.65
HTT P42858 4/20 0.63
CCR5 P51681 3/20 0.61
ALDH1A1 P00352 4/20 0.60
LMNA P02545 3/20 0.60
RAB9A P51151 1/20 0.58
PTGER1 P34995 4/20 0.56
NPC1 O15118 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
PTGDR2 Q9Y5Y4 1/20 0.54
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
HTR7 P34969 1/20 0.52
HTR6 P50406 1/20 0.52
CYP1A2 P05177 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4680227 0.87 USP28 (0.68) USP28USP25HTTCCR5ALDH1A1
SCHEMBL23275535 0.83 LRRK2 (0.54) USP28USP25HTTCCR5ALDH1A1
SCHEMBL3416114 0.83 USP28 (0.61) USP28USP25HTTCCR5ALDH1A1
SCHEMBL23275276 0.82 MEN1 (0.56) USP28USP25HTTCCR5ALDH1A1
SCHEMBL23275101 0.81 LRRK2 (0.51) USP28USP25HTTCCR5ALDH1A1
SCHEMBL22786944 0.80 USP28 (0.58) USP28USP25HTTCCR5ALDH1A1
SCHEMBL3418906 0.80 CCR5 (0.64) USP28USP25HTTCCR5ALDH1A1
SCHEMBL8807552 0.80 CCR5 (0.65) USP28USP25HTTCCR5ALDH1A1
SCHEMBL23275493 0.80 CCR5 (0.63) USP28USP25HTTCCR5ALDH1A1
SCHEMBL5305401 0.79 LMNA (0.60) ALDH1A1LMNARAB9APTGER1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7687664-B2 Carboxylic acid derivative, a salt thereof or an ester of them, and medicament comprising it EISAI R&D MANAGEMENT CO., LTD. (JP) 2010-03-30 US disclosed
EP-1394147-A1 CARBOXYLIC ACID DERIVATIVE AND MEDICINE COMPRISING SALT OR ESTER OF THE SAME Eisai Co., Ltd. (JP) 2004-03-03 EP disclosed