SCHEMBL3418973

SCHEMBL3418973

NNC(=O)c1cc(-c2cccnc2)[nH]n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.51
CYP1A2 P05177 2/20 0.51
CYP3A4 P08684 2/20 0.51
MAPT P10636 4/20 0.50
CYP2A6 P11509 2/20 0.46
CYP2B6 P20813 2/20 0.46
CYP2C9 P11712 2/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C19 P33261 1/20 0.46
HPGDS O60760 1/20 0.45
PRKAB2 O43741 1/20 0.44
PRKAG1 P54619 1/20 0.44
PRKAA2 P54646 1/20 0.44
PRKAA1 Q13131 1/20 0.44
PRKAG3 Q9UGI9 1/20 0.44
PRKAG2 Q9UGJ0 1/20 0.44
PRKAB1 Q9Y478 1/20 0.44
GSK3A P49840 1/20 0.44
GSK3B P49841 1/20 0.44
HDAC3 O15379 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL71764 0.84 EGLN3 (0.49) ALDH1A1CYP1A2CYP3A4HPGDSPRKAB2
SCHEMBL3417205 0.84 CYP3A4 (0.55) ALDH1A1CYP1A2CYP3A4CYP2A6CYP2B6
SCHEMBL3474810 0.83 ALDH1A1 (0.46) ALDH1A1CYP1A2CYP3A4MAPTCYP2A6
SCHEMBL1759178 0.82 CYP3A4 (0.57) ALDH1A1CYP1A2CYP3A4MAPTCYP2A6
Hydrochloric Acid SCHEMBL71016 0.81 CYP3A4 (0.55) ALDH1A1CYP1A2CYP3A4MAPTCYP2A6
SCHEMBL12647964 0.81 CYP1A2 (0.51) ALDH1A1CYP1A2CYP3A4CYP2A6CYP2B6
SCHEMBL12664226 0.78 CYP3A4 (0.51) ALDH1A1CYP1A2CYP3A4CYP2A6CYP2B6
SCHEMBL2818771 0.77 KMT2A (0.57) ALDH1A1CYP1A2CYP3A4MAPTCYP2C19
SCHEMBL12467859 0.76 NAMPT (0.73) CYP2C9NAMPT
SCHEMBL28425920 0.76 MAPT (0.48) CYP1A2MAPTCYP2C9CYP2C19HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107698557-B Pyridine bipyrazole acylhydrazone derivative-based fluorescent probe and preparation method and application thereof 河南理工大学 2020-10-02 CN claimed
CN-107698557-B Pyridine bipyrazole acylhydrazone derivative-based fluorescent probe and preparation method and application thereof 河南理工大学 2020-10-02 CN disclosed
EP-2593447-B1 3-PYRIDYL-HETEROARYLCARBOXAMIDE COMPOUNDS AS PESTICIDES BAYER IP GMBH (DE) 2016-08-17 EP disclosed
US-9233951-B2 Heterocyclic compounds as pesticides BAYER INTELLECTUAL PROPERTY GMBH (DE) 2016-01-12 US disclosed
US-9233951-B2 Heterocyclic compounds as pesticides BAYER INTELLECTUAL PROPERTY GMBH (DE) 2016-01-12 US disclosed
US-20120094837-A1 Novel Heterocyclic Compounds as Pesticides BAYER CROP SCIENCE AG (DE) 2012-04-19 US disclosed
US-20120094837-A1 Novel Heterocyclic Compounds as Pesticides BAYER CROP SCIENCE AG (DE) 2012-04-19 US disclosed
WO-2012007500-A2 NEW HETEROCYCLIC COMPOUNDS AS PESTICIDES BAYER CROPSCIENCE AG (DE) 2012-01-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120094837-A1 Novel Heterocyclic Compounds as Pesticides DDT, PTMS, ACHE ALDH1A1 2531/4885CYP1A2 221/4885CYP3A4 155/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.