SCHEMBL3420197

SCHEMBL3420197

CN(C)Cc1ccccc1-c1cc[c]cc1-c1cccc(-c2cccc(OCCC3CCN(C)CC3)c2)c1

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 9/20 0.52
SLC6A2 P23975 2/20 0.35
ACHE P22303 1/20 0.34
LTA4H P09960 1/20 0.34
HRH3 Q9Y5N1 3/20 0.34
KCNH2 Q12809 1/20 0.33
HTR7 P34969 1/20 0.33
CD274 Q9NZQ7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3418579 0.88 BACE1 (0.44) BACE1SLC6A2ACHEHRH3KCNH2
SCHEMBL3135802 0.77 LTA4H (0.41) BACE1LTA4HHRH3KCNH2HTR7
SCHEMBL3146491 0.77 LTA4H (0.46) BACE1LTA4HHRH3KCNH2HTR7
SCHEMBL21462366 0.71 KDM4E (0.42) ACHEHRH3
SCHEMBL21622406 0.69 BACE1 (1.00) BACE1LTA4HHRH3
SCHEMBL3133790 0.67 RAB9A (0.45) LTA4HHRH3KCNH2
SCHEMBL14426325 0.66 KDM4E (0.55) HTR7
SCHEMBL3142209 0.65 NPC1 (0.44) HRH3
SCHEMBL3425976 0.64 NOS2 (0.47) BACE1SLC6A2ACHEHRH3
SCHEMBL8265989 0.64 RAB9A (0.46) LTA4HHRH3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7666868-B2 e.g. N-Hydroxy-3-{1-[4-(1-methyl-1H-indol-5-yl)-benzenesulfonyl]-1H-pyrrol-3-yl}-acrylamide; antiproliferative, anticarcinogenic, antiinflammatory, neuroleptic agent, autoimmune disorders 4SC AG (DE) 2010-02-23 US disclosed