SCHEMBL3420535

SCHEMBL3420535

CC(C)(C)OC(=O)c1c([N+](=O)[O-])ccc(N(CCCl)CCOS(C)(=O)=O)c1[N+](=O)[O-]

nearest known ligand 0.32

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 1/20 0.32
KCNH2 Q12809 1/20 0.32
VCAM1 P19320 2/20 0.30
MAPT P10636 2/20 0.30
HTT P42858 2/20 0.30
LMNA P02545 1/20 0.30
THRB P10828 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
GPR55 Q9Y2T6 1/20 0.30
MET P08581 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2974168 0.87 KDM4E (0.35) HCAR3KCNH2MAPT
SCHEMBL3417440 0.86 NSD2 (0.39) HCAR3VCAM1MAPTHTT
SCHEMBL2969505 0.85 VCAM1 (0.39) HCAR3KCNH2VCAM1MAPTHTT
SCHEMBL2976494 0.82 HCAR3 (0.42) HCAR3KCNH2HTT
SCHEMBL13202988 0.81 KCNH2 (0.37) HCAR3KCNH2VCAM1MAPT
SCHEMBL2977189 0.81 ALDH1A1 (0.37) KCNH2MAPTLMNATHRBNPSR1
SCHEMBL5675133 0.81
SCHEMBL3421976 0.80 VCAM1 (0.35) HCAR3KCNH2VCAM1MAPTHTT
SCHEMBL2977431 0.79 ALDH1A1 (0.34) KCNH2
SCHEMBL3585555 0.78 ALDH1A1 (0.36) KCNH2LMNATHRBNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100121091-A1 Processes of preparing asymmetric dinitrobenzamide mustard compounds, intermediate compounds useful therein and products obtained therefrom AUCKLAND UNISERVICES LIMITED (NZ) 2010-05-13 US disclosed
EP-2059499-A1 PROCESSES OF PREPARING ASYMMETRIC DINITROBENZAMIDE MUSTARD COMPOUNDS, INTERMEDIATE COMPOUNDS USEFUL THEREIN AND PRODUCTS OBTAINED THEREFROM Auckland Uniservices Limited (NZ) 2009-05-20 EP disclosed
WO-2008030112-A1 PROCESSES OF PREPARING ASYMMETRIC DINITROBENZAMIDE MUSTARD COMPOUNDS, INTERMEDIATE COMPOUNDS USEFUL THEREIN AND PRODUCTS OBTAINED THEREFROM AUCKLAND UNISERVICES LIMITED (NZ) 2008-03-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100121091-A1 Processes of preparing asymmetric dinitrobenzamide mustard compounds, intermediate compounds useful therein and products obtained therefrom HRH2, HRH4, H1-2 HCAR3 275/4885KCNH2 291/4885VCAM1 4320/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.