SCHEMBL3420564

SCHEMBL3420564

COc1c(C)cc(-c2ccc[nH]c2=O)cc1C1C[C@@H]1c1ccc(NS(C)(=O)=O)cc1

nearest known ligand 0.79

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.79
KDM1A O60341 8/20 0.41
MAOA P21397 3/20 0.37
MAOB P27338 1/20 0.37
NR3C1 P04150 6/20 0.36
PGR P06401 5/20 0.36
NR3C2 P08235 5/20 0.36
BRD4 O60885 3/20 0.36
EP300 Q09472 2/20 0.36
AR P10275 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3422415 1.00 CYP3A4 (0.79) CYP3A4KDM1AMAOAMAOBNR3C1
SCHEMBL2112475 0.89 CYP3A4 (1.00) CYP3A4KDM1AMAOAMAOBNR3C1
SCHEMBL725581 0.89 CYP3A4 (1.00) CYP3A4KDM1AMAOAMAOBNR3C1
SCHEMBL2111363 0.89 CYP3A4 (1.00) CYP3A4KDM1AMAOAMAOBNR3C1
SCHEMBL724765 0.88 CYP3A4 (0.75) CYP3A4KDM1AMAOAMAOBNR3C1
SCHEMBL3421761 0.82 CYP3A4 (0.63) CYP3A4KDM1AMAOAMAOBNR3C1
SCHEMBL2111644 0.78 CYP3A4 (0.69) CYP3A4KDM1AMAOAMAOBNR3C2
SCHEMBL3423335 0.77 CYP3A4 (0.57) CYP3A4KDM1ANR3C1PGRNR3C2
SCHEMBL726323 0.74 CYP3A4 (0.64) CYP3A4KDM1ANR3C2BRD4EP300
SCHEMBL3478670 0.73 CYP3A4 (0.56) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8158803-B2 Heterocyclic antiviral compounds ROCHE PALO ALTO LLC (US) 2012-04-17 US disclosed
US-20100272677-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS LEE EUN KYUNG 2010-10-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100272677-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS POLR2A, EIF2AK2, RRM2B CYP3A4 417/4885KDM1A 1567/4885MAOA 733/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.