SCHEMBL3421702

SCHEMBL3421702

O=C(NC1CC1)C1CNCCC1(O)c1ccc(F)c(F)c1

nearest known ligand 0.52

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
REN P00797 20/20 0.52
KCNH2 Q12809 20/20 0.52
CYP3A4 P08684 6/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3102591 0.69 REN (1.00) RENKCNH2CYP3A4
SCHEMBL3102603 0.69 REN (1.00) RENKCNH2CYP3A4
SCHEMBL533858 0.68 REN (0.46) RENKCNH2CYP3A4
SCHEMBL7004831 0.66 REN (0.42) RENKCNH2CYP3A4
SCHEMBL533971 0.65 DRD2 (0.59) RENKCNH2CYP3A4
Hydrochloric Acid SCHEMBL22616883 0.63 DRD2 (0.58) RENKCNH2CYP3A4
SCHEMBL6966294 0.63 GHSR (0.43)
SCHEMBL3107459 0.62 DRD2 (0.47) RENKCNH2CYP3A4
SCHEMBL651950 0.62 DRD2 (0.41) RENKCNH2
SCHEMBL5169982 0.62 CYP2C19 (0.44) RENKCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2229363-A1 RENIN INHIBITORS Merck Frosst Canada Ltd. (CA) 2010-09-22 EP disclosed
WO-2009070869-A1 RENIN INHIBITORS MERCK FROSST CANADA LTD. (CA) 2009-06-11 WO disclosed