SCHEMBL3427816

SCHEMBL3427816

Cc1cc(C)cc(N2CC=CN2)c1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.35
MAPT P10636 2/20 0.34
ALDH1A1 P00352 1/20 0.34
HSP90AA1 P07900 1/20 0.33
CCR6 P51684 1/20 0.33
HPGD P15428 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
KDM4E B2RXH2 1/20 0.31
NOTUM Q6P988 1/20 0.31
HCAR1 Q9BXC0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11401376 0.75
SCHEMBL12354590 0.67 BPTF (0.33)
SCHEMBL28030094 0.62 ADRB1 (0.39) NPSR1MAPTALDH1A1HSP90AA1CCR6
SCHEMBL24197603 0.60 ALDH1A1 (0.40) ALDH1A1
SCHEMBL28300826 0.59 ALDH1A1 (0.50) NPSR1MAPTALDH1A1HSP90AA1CCR6
SCHEMBL341533 0.58 ALDH1A1 (0.67) ALDH1A1HSP90AA1CCR6
SCHEMBL26115 0.58
SCHEMBL1138607 0.57 ADRB1 (0.66) MAPTALDH1A1
SCHEMBL4760153 0.56 ALDH1A1 (0.40) NPSR1MAPTALDH1A1HSP90AA1CCR6
SCHEMBL3543974 0.56 MAPT (0.50) NPSR1MAPTALDH1A1HSP90AA1CCR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101965350-A Novel pyrazolo [3,4-d ] pyrimidine derivatives as anticancer agents NATCO PHARMA LTD 2011-02-02 CN disclosed
EP-2247596-A2 NOVEL PYRAZOLO [3, 4 -D] PYRIMIDINE DERIVATIVES AS ANTI -CANCER AGENTS Natco Pharma Limited (IN) 2010-11-10 EP disclosed
WO-2009098715-A2 NOVEL PYRAZOLO [3, 4 -D] PYRIMIDINE DERIVATIVES AS ANTI -CANCER AGENTS NATCO PHARMA LIMITED (IN) 2009-08-13 WO disclosed