SCHEMBL3428079

SCHEMBL3428079

COc1ccc2ncc(F)c(CNC3CN(C[C@H]4COC(=O)N4c4ccc5c(c4)NC(=O)CO5)C3)c2c1

nearest known ligand 0.51

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 9/20 0.43
SLC2A1 P11166 1/20 0.40
KCNQ1 P51787 1/20 0.40
CACNA1C Q13936 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3425401 0.88 KCNH2 (0.54) KCNH2
SCHEMBL3423438 0.87 KCNH2 (0.53) KCNH2KCNQ1CACNA1C
SCHEMBL633085 0.87 KCNH2 (0.43) KCNH2SLC2A1KCNQ1CACNA1C
SCHEMBL633042 0.87 KCNH2 (0.43) KCNH2SLC2A1KCNQ1CACNA1C
SCHEMBL3427490 0.84 KCNH2 (0.45) KCNH2KCNQ1CACNA1C
SCHEMBL3396541 0.79 KCNH2 (0.41) KCNH2KCNQ1CACNA1C
SCHEMBL3668001 0.78 DRD4 (0.40) KCNH2
SCHEMBL3419619 0.77 KCNH2 (0.44) KCNH2
SCHEMBL592146 0.76 GRM2 (0.39) KCNH2
SCHEMBL590312 0.76 GRM2 (0.39) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2245028-A1 5-AMINOCYCLYLMETHYL-OXAZOLIDIN-2-ONE DERIVATIVES Actelion Pharmaceuticals Ltd. (CH) 2010-11-03 EP disclosed
WO-2009077989-A1 5-AMINOCYCLYLMETHYL-OXAZOLIDIN-2-ONE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2009-06-25 WO disclosed