SCHEMBL3431056

SCHEMBL3431056

c1ccc(CSNc2ccccc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 5/20 0.40
TDP1 Q9NUW8 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
LMNA P02545 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
PTGS2 P35354 1/20 0.40
NOS3 P29474 1/20 0.40
NOS1 P29475 1/20 0.40
NOS2 P35228 1/20 0.40
HSD17B10 Q99714 2/20 0.39
POLB P06746 1/20 0.39
MAOB P27338 1/20 0.39
METAP2 P50579 1/20 0.39
METAP1 P53582 1/20 0.39
CTSL P07711 1/20 0.38
CTSB P07858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28116299 0.81 NPSR1 (0.52) LMNACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL22700102 0.81 KDM4E (0.52) TDP1LMNACYP3A4POLBMAOB
SCHEMBL14776233 0.77 TDP1 (0.46) IDO1TDP1L3MBTL1LMNACYP1A2
SCHEMBL11265077 0.77 KCNH3 (0.57) LMNAMETAP2METAP1
SCHEMBL7072380 0.73 ALDH1A1 (0.42) IDO1TDP1L3MBTL1LMNACYP1A2
SCHEMBL18962146 0.73 CYP3A4 (0.46) IDO1L3MBTL1LMNACYP1A2CYP3A4
SCHEMBL8534443 0.73 IDO1 (0.42) IDO1TDP1CYP1A2CYP3A4CYP2D6
SCHEMBL6676668 0.73 TDP1 (0.42) IDO1TDP1L3MBTL1LMNACYP1A2
SCHEMBL9577412 0.73 IDO1 (0.41) IDO1TDP1CYP1A2CYP3A4CYP2D6
SCHEMBL31161041 0.73 SMN1; SMN2 (0.44) TDP1L3MBTL1LMNACYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105646396-B A kind of synthetic method of benzothiazole derivant 上海应用技术学院 2018-09-14 CN claimed
WO-2010068296-A1 PIPERAZINE CARBOXAMIDINES AS ANTIMICROBIAL AGENTS STIEFEL LABORATORIES, INC. (US) 2010-06-17 WO disclosed
US-5116851-A Administering antiischemic and antiarrhythmia agents E. R. SQUIBB & SONS, INC. (US) 1992-05-26 US disclosed
EP-0453658-A2 Use of substituted anilides and sulfonamides in the treatment of cardiovascular diseases E.R. SQUIBB & SONS, INC. (US) 1991-10-30 EP disclosed