SCHEMBL3431395

SCHEMBL3431395

O=c1[nH]c2cc(-c3ccc(OC(F)(F)F)cc3)ccc2nc1CCc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.56
NPC1 O15118 1/20 0.56
RAB9A P51151 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
TRPV1 Q8NER1 4/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
GAA P10253 1/20 0.43
HPGD P15428 1/20 0.43
HSD17B10 Q99714 1/20 0.43
PDE10A Q9Y233 1/20 0.41
DAO P14920 1/20 0.41
RUNX1 Q01196 2/20 0.41
CBFB Q13951 1/20 0.41
CACNA1B Q00975 1/20 0.41
GPR84 Q9NQS5 1/20 0.40
CHEK2 O96017 1/20 0.40
EGLN1 Q9GZT9 2/20 0.39
HDAC6 Q9UBN7 1/20 0.39
MEN1 O00255 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3377915 0.79 CYP1A2 (0.45) SMN1; SMN2ALDH1A1HPGDHSD17B10HDAC6
SCHEMBL3476576 0.77 TRPV1 (0.50) TRPV1RUNX1CBFBCACNA1BCHEK2
SCHEMBL3474853 0.76 PDE4A (0.43) KDM4EALDH1A1HPGDHSD17B10POLB
Hydrochloric Acid SCHEMBL11903522 0.74 PDE10A (0.67) HTTNPC1RAB9ASMN1; SMN2TRPV1
SCHEMBL3430623 0.73 FFAR1 (0.43) HTTKDM4EALDH1A1GAAHPGD
SCHEMBL3431393 0.72 SERPINE1 (0.43) HDAC6SERPINE1
Hydrochloric Acid SCHEMBL11903596 0.69 GAA (0.61) TRPV1KDM4EGAAPDE10ARUNX1
Hydrochloric Acid SCHEMBL11903518 0.67 RAB9A (0.56) HTTNPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL5952465 0.67 RUNX1 (0.49) TRPV1PDE10ARUNX1CBFBCHEK2
SCHEMBL11903481 0.67 TRPV1 (0.72) HTTNPC1RAB9ASMN1; SMN2TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010053757-A1 2 -OXOQUINOXALIN BLOCKERS OF THE LATE SODIUM CHANNEL GILEAD PALO ALTO, INC. (US) 2010-05-14 WO claimed