SCHEMBL343298

SCHEMBL343298

Nc1ccc(Cl)cc1C(=O)c1ccc(Cl)nc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RECQL P46063 1/20 0.53
NAPRT Q6XQN6 1/20 0.49
CCR9 P51686 3/20 0.47
FADS1 O60427 1/20 0.44
MAPT P10636 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
KCNQ3 O43525 2/20 0.43
KCNQ2 O43526 2/20 0.43
KCNE1 P15382 2/20 0.43
KCNQ1 P51787 2/20 0.43
GFER P55789 1/20 0.43
KMT2A Q03164 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
GCK P35557 1/20 0.43
EGFR P00533 1/20 0.43
ALDH1A1 P00352 1/20 0.42
POLB P06746 1/20 0.42
NOS2 P35228 1/20 0.42
DYRK3 O43781 1/20 0.42
CCNA2 P20248 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL343308 0.85 CCR9 (0.55) RECQLCCR9FADS1MAPTTDP1
SCHEMBL6351799 0.82 RECQL (0.64) RECQLFADS1MAPTTDP1GFER
SCHEMBL15308437 0.82 NAPRT (0.49) NAPRTCCR9MAPTKCNQ3KCNQ2
SCHEMBL10633292 0.81 SRD5A2 (0.59) NAPRTCCR9MAPTKCNQ3KCNQ2
SCHEMBL343984 0.80 ALDH1A1 (0.50) NAPRTCCR9MAPTKMT2ASMN1; SMN2
SCHEMBL12653273 0.79 RECQL (0.60) RECQLFADS1MAPTTDP1GFER
SCHEMBL342198 0.79 RECQL (0.53) RECQLCCR9FADS1MAPTTDP1
SCHEMBL344032 0.79 RECQL (0.53) RECQLCCR9FADS1MAPTTDP1
SCHEMBL28232 0.79 CCR9 (0.58) RECQLCCR9TDP1KMT2ASMN1; SMN2
SCHEMBL9540049 0.78 RECQL (0.79) RECQLFADS1TDP1GFERKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 55 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10364240-B2 Aryl sulfonamides ChemoCentryx. Inc. (US) 2019-07-30 US disclosed
US-10364240-B2 Aryl sulfonamides ChemoCentryx. Inc. (US) 2019-07-30 US disclosed
US-9890148-B2 Aryl sulfonamides CHEMOCENTRYX, INC. (US) 2018-02-13 US disclosed
US-9890148-B2 Aryl sulfonamides CHEMOCENTRYX, INC. (US) 2018-02-13 US disclosed
US-20170369483-A1 ARYL SULFONAMIDES CHEMOCENTRYX, INC. (US) 2017-12-28 US disclosed
US-20150080351-A1 ARYL SULFONAMIDES CHEMOCENTRYX, INC. 2015-03-19 US disclosed
US-20150080351-A1 ARYL SULFONAMIDES CHEMOCENTRYX, INC. 2015-03-19 US disclosed
US-20150080351-A1 ARYL SULFONAMIDES CHEMOCENTRYX, INC. 2015-03-19 US disclosed
EP-1798223-B2 Aryl sulfonamides CHEMOCENTRYX INC (US) 2014-07-30 EP disclosed
US-20130267492-A1 ARYL SULFONAMIDES CHEMOCENTRYX, INC. (US) 2013-10-10 US disclosed
US-20060111351-A1 Aryl sulfonamides CHEMOCENTRYX, INC. 2006-05-25 US disclosed
CN-1711257-A Aryl sulfonamides CHEMOCENTRYX (US) 2005-12-21 CN disclosed
WO-2005112925-A1 ARYL SULFONAMIDES CHEMOCENTRYX (US) 2005-12-01 WO disclosed
US-6939885-B2 Aryl sulfonamides CHEMOCENTRYX (US) 2005-09-06 US disclosed
EP-1562940-A2 ARYL SULFONAMIDES ChemoCentryx Inc (US) 2005-08-17 EP disclosed
US-20050165067-A1 Aryl sulfonamides CHEMOCENTRYX 2005-07-28 US disclosed
US-20050137193-A1 Aryl sulfonamides CHEMOCENTREYX 2005-06-23 US disclosed
WO-2005051381-A1 Substituted urea-octatydroindols as antagonists of melanin concentrating hormone receptor 1 (MCH1R) BIOVITRUM AB (SE) 2005-06-09 WO disclosed
US-20040171654-A1 Aryl sulfonamides CHEMOCENTRYX, INC. 2004-09-02 US disclosed
WO-2004046092-A2 ARYL SULFONAMIDES CHEMOCENTRYX (US) 2004-06-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050137193-A1 Aryl sulfonamides CCR9, CCR1, CCR2 RECQL 4746/4885NAPRT 791/4885CCR9 1/4885
US-10364240-B2 Aryl sulfonamides CCR9, CCR1, CCR2 RECQL 4746/4885NAPRT 791/4885CCR9 1/4885
US-20060111351-A1 Aryl sulfonamides CCR9, CCR1, CCR2 RECQL 4746/4885NAPRT 791/4885CCR9 1/4885
US-20170369483-A1 ARYL SULFONAMIDES CCR9, CCR1, CCR2 RECQL 4746/4885NAPRT 791/4885CCR9 1/4885
US-20150080351-A1 ARYL SULFONAMIDES CCR9, CCR1, CCR2 RECQL 4746/4885NAPRT 791/4885CCR9 1/4885
US-20040171654-A1 Aryl sulfonamides CCR9, CCR1, CCR2 RECQL 4746/4885NAPRT 791/4885CCR9 1/4885
US-20050165067-A1 Aryl sulfonamides CCR9, CCR1, CCR2 RECQL 4746/4885NAPRT 791/4885CCR9 1/4885
US-20130267492-A1 ARYL SULFONAMIDES CCR9, CCR1, CCR2 RECQL 4746/4885NAPRT 791/4885CCR9 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.