SCHEMBL3433332

SCHEMBL3433332

COC(=O)c1ccc2c(c1)c(CC1COCCN1)cn2C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 2/20 0.40
PARG Q86W56 1/20 0.40
ALDH1A1 P00352 3/20 0.39
PDGFRB P09619 2/20 0.39
KDR P35968 2/20 0.39
PIK3C2A O00443 1/20 0.39
PIK3C2B O00750 1/20 0.39
CNR1 P21554 1/20 0.38
IDH1 O75874 1/20 0.38
SCARB1 Q8WTV0 1/20 0.38
MAPK1 P28482 1/20 0.36
BRD4 O60885 1/20 0.36
CREBBP Q92793 1/20 0.36
NQO2 P16083 1/20 0.36
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36
CCNT1 O60563 1/20 0.36
CCNA2 P20248 1/20 0.36
CDK2 P24941 1/20 0.36
GSK3A P49840 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL945731 1.00 CNR2 (0.40) CNR2PARGALDH1A1PDGFRBKDR
SCHEMBL945617 0.80 GPR84 (0.54) PDGFRB
SCHEMBL1855927 0.78 NPC1 (0.57) ALDH1A1PDGFRBMAPK1CDK2
SCHEMBL947139 0.78 SLC6A4 (0.45) CNR2PARGALDH1A1PDGFRBPIK3C2A
SCHEMBL3433438 0.77 CNR2 (0.45) CNR2PARGCNR1CCNT1CCNA2
SCHEMBL3433442 0.77 CNR2 (0.45) CNR2PARGCNR1CCNT1CCNA2
SCHEMBL944734 0.77 GPR84 (0.48) ALDH1A1
SCHEMBL944759 0.76 PIK3C2A (0.43) CNR2ALDH1A1PDGFRBPIK3C2APIK3C2B
SCHEMBL3434033 0.72 HTR1A (0.37) PARGALDH1A1PIK3C2APIK3C2B
SCHEMBL3433906 0.72 PIK3C2A (0.41) ALDH1A1PIK3C2APIK3C2BMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2170906-B1 FUSED THIAZOLE DERIVATIVES AS KINASE INHIBITORS UCB PHARMA SA (BE) 2013-04-03 EP disclosed
WO-2010146351-A1 INDOLYLMETHYL-MORPHOLINE DERIVATIVES AS KINASE INHIBITORS UCB PHARMA S.A. (BE) 2010-12-23 WO disclosed