SCHEMBL3434696

SCHEMBL3434696

C=CCC(CC=C)(c1ccc([N+](=O)[O-])cc1)P(=O)(O)O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
MAPT P10636 3/20 0.42
KDM4E B2RXH2 1/20 0.42
LMNA P02545 1/20 0.42
HTT P42858 1/20 0.42
AKR1C3 P42330 1/20 0.42
CA1 P00915 3/20 0.41
CA2 P00918 3/20 0.41
CES1 P23141 2/20 0.41
CES2 O00748 1/20 0.41
CYP2C19 P33261 1/20 0.40
POLB P06746 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
CA12 O43570 2/20 0.39
MMP2 P08253 2/20 0.39
MMP9 P14780 1/20 0.39
MMP8 P22894 1/20 0.39
MMP14 P50281 1/20 0.39
TGM2 P21980 1/20 0.39
PTPRC P08575 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL78562 0.80 ALDH1A1 (0.51) ALDH1A1MAPTLMNAAKR1C3CA1
SCHEMBL2052519 0.78 FDPS (0.43) ALDH1A1MAPTKDM4ELMNAHTT
SCHEMBL2033791 0.75 ALDH1A1 (0.47) ALDH1A1MAPTLMNAAKR1C3CA1
SCHEMBL8020613 0.74 ALDH1A1 (0.63) ALDH1A1MAPTKDM4ELMNAHTT
SCHEMBL10685573 0.74 CYP2C19 (0.50) ALDH1A1MAPTKDM4ELMNAHTT
SCHEMBL830832 0.72 CYP2C19 (0.42) ALDH1A1MAPTKDM4ELMNAHTT
SCHEMBL5897358 0.72 CA1 (0.50) AKR1C3CA1CA2CES1CES2
Allyl Alcohol SCHEMBL28052693 0.70 TSHR (0.55) ALDH1A1MAPTKDM4ELMNAHTT
SCHEMBL2030739 0.70 CA1 (0.49) ALDH1A1AKR1C3CA1CA2CES1
SCHEMBL2637314 0.70 PTPRC (0.51) ALDH1A1MAPTKDM4ELMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1542970-B1 PYRROLIDONE DERIVATIVES AS MAOB INHIBITORS HOFFMANN LA ROCHE (CH) 2010-06-30 EP disclosed
US-7151111-B2 4-pyrrolidino-phenyl-benzyl ether derivatives HOFFMANN-LA ROCHE INC. (US) 2006-12-19 US disclosed
EP-1542970-A1 PYRROLIDONE DERIVATIVES AS MAOB INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2005-06-22 EP disclosed
US-20040116707-A1 4-Pyrrolidino-phenyl-benzyl ether derivatives HOFFMANN-LA ROCHE INC. 2004-06-17 US disclosed
WO-2004026825-A1 PYRROLIDONE DERIVATIVES AS MAOB INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2004-04-01 WO disclosed