SCHEMBL5897358

SCHEMBL5897358

O=[N+]([O-])c1ccc(C(O)(P(=O)(O)O)P(=O)(O)O)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.50
CA2 P00918 4/20 0.50
CES1 P23141 2/20 0.50
CES2 O00748 1/20 0.50
PTPRC P08575 1/20 0.49
CA12 O43570 2/20 0.46
MMP2 P08253 2/20 0.46
AKR1C3 P42330 1/20 0.46
MMP9 P14780 1/20 0.46
MMP8 P22894 1/20 0.46
MMP14 P50281 1/20 0.46
HSD11B1 P28845 1/20 0.44
CYP19A1 P11511 1/20 0.44
CA9 Q16790 2/20 0.43
CA5A P35218 1/20 0.43
CA14 Q9ULX7 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
MEN1 O00255 1/20 0.42
POLB P06746 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16253828 0.81 PGK1 (0.52)
SCHEMBL2030739 0.79 CA1 (0.49) CA1CA2CES1CES2PTPRC
SCHEMBL3230183 0.79 PTPRC (0.51) CA1CA2CES1CES2PTPRC
SCHEMBL2637314 0.79 PTPRC (0.51) CA1CA2CES1CES2PTPRC
SCHEMBL2636706 0.79 PGK1 (0.67) CA1CA2CES1CES2HSD11B1
Phosphoric Acid SCHEMBL28639141 0.79 CA1 (0.65) CA1CA2CES1CES2CA12
SCHEMBL78562 0.75 ALDH1A1 (0.51) CA1CA2CES1CES2PTPRC
SCHEMBL11029750 0.74 PTPRC (0.43) CA1CA2CES1CES2PTPRC
SCHEMBL1023276 0.74 HSD11B1 (0.60) CA1CA2CES1HSD11B1CYP19A1
SCHEMBL11026039 0.74 CES1 (0.54) CA1CA2CES1CES2HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7005533-B2 Bisphosphonate derivatives, their preparations and uses UNIVERSITE PARIS 13 (FR) 2006-02-28 US disclosed
US-20040266735-A1 Bisphosphonate derivatives, their preparations and uses UNIVERSITE PARIS 13 2004-12-30 US disclosed
US-20030036537-A1 Bisphosphonate derivatives, their preparations and uses UNIVERSITE PARIS, 13 (FR) 2003-02-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030036537-A1 Bisphosphonate derivatives, their preparations and uses BPGM, PPIP5K2, PTEN CA1 3133/4885CA2 1168/4885CES1 2004/4885
US-20040266735-A1 Bisphosphonate derivatives, their preparations and uses BPGM, PPIP5K2, PTEN CA1 3133/4885CA2 1168/4885CES1 2004/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.