SCHEMBL3435446

SCHEMBL3435446

O=C(O)C(c1cccc(-c2ccccc2)c1)C(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTPN5 P54829 6/20 0.46
RXRA P19793 1/20 0.45
RXRB P28702 1/20 0.45
RXRG P48443 1/20 0.45
PTPN1 P18031 2/20 0.44
KMO O15229 1/20 0.42
HDAC4 P56524 1/20 0.41
PTGS2 P35354 1/20 0.41
APP P05067 1/20 0.40
CTSA P10619 1/20 0.40
MGLL Q99685 1/20 0.40
CYP2D6 P10635 1/20 0.39
SRC P12931 1/20 0.39
CTSL P07711 1/20 0.39
CTSS P25774 1/20 0.39
CTSK P43235 1/20 0.39
ABHD6 Q9BV23 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL195532 0.83 SRC (0.50) HDAC4CYP2D6SRC
SCHEMBL4026079 0.83 SRC (0.50) HDAC4CYP2D6SRC
SCHEMBL7955519 0.83 SRC (0.50) HDAC4CYP2D6SRC
Hydrochloric Acid SCHEMBL2529822 0.81 SRC (0.48) CYP2D6SRC
SCHEMBL29773675 0.81 SRC (0.48) HDAC4CYP2D6SRC
SCHEMBL28789627 0.81 HDAC4 (0.49) HDAC4
Methyl Alcohol SCHEMBL5139174 0.80 SRC (0.46) CYP2D6SRC
SCHEMBL5574337 0.79 CES2 (0.54)
SCHEMBL28829348 0.79 MEN1 (0.48)
SCHEMBL11543519 0.79 PTGS1 (0.60) HDAC4MGLLCYP2D6ABHD6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2257524-A1 N,N-DISUBSTITUTED AMINOALKYLBIPHENYL ANTAGONISTS OF PROSTAGLANDIN D2 RECEPTORS Amira Pharmaceuticals, Inc. (US) 2010-12-08 EP disclosed
WO-2009099902-A1 N,N-DISUBSTITUTED AMINOALKYLBIPHENYL ANTAGONISTS OF PROSTAGLANDIN D2 RECEPTORS AMIRA PHARMACEUTICALS, INC. (US) 2009-08-13 WO disclosed