Gentisic Acid

Gentisic Acid

SCHEMBL344389

O=C(O)c1cc(O)ccc1O.[KH]

nearest known ligand 0.95

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.95
CA2 P00918 4/20 0.95
CA12 O43570 3/20 0.95
CA7 P43166 3/20 0.95
CA9 Q16790 3/20 0.95
CA14 Q9ULX7 3/20 0.95
PTGS2 P35354 3/20 0.95
ALOX5 P09917 1/20 0.95
ALDH1A1 P00352 3/20 0.64
TSHR P16473 1/20 0.64
MEN1 O00255 2/20 0.59
KDR P35968 2/20 0.59
KMT2A Q03164 2/20 0.59
HSD17B10 Q99714 2/20 0.59
TDP1 Q9NUW8 2/20 0.59
KDM4E B2RXH2 1/20 0.59
TNF P01375 1/20 0.59
CYP3A4 P08684 1/20 0.59
HSPD1 P10809 1/20 0.59
THRB P10828 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Gentisic Acid SCHEMBL3690 0.98 CA1 (1.00) CA1CA2CA12CA7CA9
Gentisic Acid SCHEMBL30233582 0.98 CA1 (1.00) CA1CA2CA12CA7CA9
Gentisic Acid SCHEMBL2053863 0.98 CA1 (1.00) CA1CA2CA12CA7CA9
Gentisic Acid SCHEMBL29349919 0.98 CA1 (1.00) CA1CA2CA12CA7CA9
Gentisic Acid SCHEMBL8922036 0.95 CA1 (0.95) CA1CA2CA12CA7CA9
Gentisic Acid SCHEMBL450480 0.95 CA1 (0.95) CA1CA2CA12CA7CA9
Gentisic Acid SCHEMBL10975219 0.95 CA1 (0.95) CA1CA2CA12CA7CA9
Gentisic Acid SCHEMBL10978035 0.95 CA1 (0.95) CA1CA2CA12CA7CA9
Gentisic Acid SCHEMBL3981503 0.95 CA1 (0.95) CA1CA2CA12CA7CA9
Gentisic Acid SCHEMBL10980548 0.95 CA1 (0.95) CA1CA2CA12CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 54 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012114342-A1 FLUMAZENIL COMPLEXES, COMPOSITIONS COMPRISING SAME AND USES THEREOF COERULEUS LTD. (IL) 2012-08-30 WO claimed
CN-116410727-A Dilution thickening type surfactant spherical micelle super-concentrated dispersion system, and preparation method and application thereof 武汉大学 2023-07-11 CN disclosed
US-20190192474-A1 Use Of 2,5-Dihydroxybenzene Compounds And Derivatives For The Treatment Of Skin Cancer AmDerma Pharmaceuticals, LLC 2019-06-27 US disclosed
US-20190192473-A1 Use Of 2,5-Dihydroxybenzene Compounds And Derivatives For The Treatment Of Rosacea AmDerma Pharmaceuticals, LLC 2019-06-27 US disclosed
US-10278940-B2 Use of 2,5-dihydroxybenzene compounds and derivatives for the treatment of skin cancer AmDerma Pharmaceuticals, LLC (US) 2019-05-07 US disclosed
US-10278941-B2 Use of 2,5-dihydroxybenzene compounds and derivatives for the treatment of glioma AmDerma Pharmaceuticals, LLC (US) 2019-05-07 US disclosed
US-20180028484-A1 Use Of 2,5-Dihydroxybenzene Compounds And Derivatives For The Treatment Of Rosacea AmDerma Pharmaceuticals, LLC 2018-02-01 US disclosed
US-9592216-B2 Use of 2,5-dihydroxybenzene compounds and derivatives for the treatment of rosacea AmDerma Pharmaceuticals, LLC (US) 2017-03-14 US disclosed
US-20170065547-A1 Use Of 2,5-Dihydroxybenzene Compounds And Derivatives For The Treatment Of Skin Cancer ACTION MEDICINES, S.L. (ES) 2017-03-09 US disclosed
US-9585893-B2 Flumazenil complexes, compositions comprising same and uses thereof COERULEUS LTD. (IL) 2017-03-07 US disclosed
WO-2008020039-A2 2,5-DIHYDROXYBENZENE COMPOUNDS FOR TREATING CANCERS AND HEMATOLOGICAL DYSCRASIAS ACTION MEDICINES, S.L. (ES) 2008-02-21 WO disclosed
WO-2008020030-A1 2,5-DIHYDROXYBENZENE COMPOUNDS FOR THE TREATMENT OF PSORIASIS ACTION MEDICINES, S.L. (ES) 2008-02-21 WO disclosed
WO-2008020027-A2 2,5-DIHYDROXYBENZENE COMPOUNDS FOR THE TREATMENT OF SKIN CANCER ACTION MEDICINES, S.L. (ES) 2008-02-21 WO disclosed
WO-2008020028-A1 2,5 DIHYDROXYBENZENE COMPOUNDS FOR THE TREATMENT OF ROSACEA ACTION MEDICINES, S.L. (ES) 2008-02-21 WO disclosed
WO-2008020031-A1 USE OF 2,5-DIHYDROXYBENZENE DERIVATIVES FOR THE TREATMENT OF ANGIOGENIC DISEASES ACTION MEDICINES, S.L. (ES) 2008-02-21 WO disclosed
WO-2008020040-A2 2,5-DIHYDROXYBENZENE COMPOUNDS FOR THE TREATMENT OF FIBROSIS ACTION MEDICINES, S.L. (ES) 2008-02-21 WO disclosed
US-4497744-A Gentisic acid salts as radiographic scanning agent stabilizers MALLINCKRODT, INC. (US) 1985-02-05 US disclosed
EP-0004684-B1 STABILIZED RADIOGRAPHIC SCANNING AGENTS AND METHOD FOR PREPARING THEM THE PROCTER & GAMBLE COMPANY (US) 1981-09-16 EP disclosed
US-4233284-A GENESTIC ACID, SALT OR ESTER THEREOF IN COMBINATION WITH A PERTECHNETATE REDUCING AGENT BECOMES LOCALIZED IN SPECIFIC BODY ORGANS OR BONES THE PROCTER & GAMBLE COMPANY (US) 1980-11-11 US disclosed
EP-0004684-A2 Stabilized radiographic scanning agents and method for preparing them THE PROCTER & GAMBLE COMPANY (US) 1979-10-17 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190192473-A1 Use Of 2,5-Dihydroxybenzene Compounds And Derivatives For The Treatment Of Rosacea CYP8B1, CYP1B1, CYP26B1 CA1 2993/4885CA2 899/4885CA12 1207/4885
US-10278940-B2 Use of 2,5-dihydroxybenzene compounds and derivatives for the treatment of skin cancer CYP8B1, CYP26B1, CYP24A1 CA1 1782/4885CA2 463/4885CA12 431/4885
US-20170065547-A1 Use Of 2,5-Dihydroxybenzene Compounds And Derivatives For The Treatment Of Skin Cancer CYP8B1, CYP26B1, CYP24A1 CA1 1782/4885CA2 463/4885CA12 431/4885
US-20190192474-A1 Use Of 2,5-Dihydroxybenzene Compounds And Derivatives For The Treatment Of Skin Cancer CYP8B1, CYP26B1, CYP24A1 CA1 1782/4885CA2 463/4885CA12 431/4885
US-20180028484-A1 Use Of 2,5-Dihydroxybenzene Compounds And Derivatives For The Treatment Of Rosacea CYP8B1, CYP1B1, CYP26B1 CA1 2993/4885CA2 899/4885CA12 1207/4885
US-10278941-B2 Use of 2,5-dihydroxybenzene compounds and derivatives for the treatment of glioma ALDH1A2, IDH3A, IDH3B CA1 312/4885CA2 340/4885CA12 180/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.