Nitroarginine

Nitroarginine

SCHEMBL345312

N=C(NCCC[C@H](N)C(=O)O)N[N+](=O)[O-]

nearest known ligand 0.48

Full drug profile on Sugi Atlas →

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 4/20 0.48
NOS3 P29474 2/20 0.48
NOS2 P35228 2/20 0.48
OTC P00480 1/20 0.47
DDAH1 O94760 1/20 0.41
GSR P00390 1/20 0.40
ARG1 P05089 3/20 0.37
ARG2 P78540 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Nitroarginine SCHEMBL28365071 1.00 NOS1 (0.48) NOS1NOS3NOS2OTCDDAH1
Nitroarginine SCHEMBL881062 1.00 NOS1 (0.48) NOS1NOS3NOS2OTCDDAH1
SCHEMBL607060 0.88 NOS1 (0.46) NOS1NOS3NOS2OTCDDAH1
SCHEMBL5983469 0.88 NOS1 (0.46) NOS1NOS3NOS2OTCDDAH1
L-Name SCHEMBL3034749 0.84 NOS1 (0.41) NOS1NOS3NOS2OTC
L-Name SCHEMBL14751988 0.84 NOS1 (0.41) NOS1NOS3NOS2OTC
L-Name SCHEMBL25310005 0.83 NOS1 (0.40) NOS1NOS3NOS2OTC
L-Name SCHEMBL18812631 0.83 NOS1 (0.40) NOS1NOS3NOS2OTC
SCHEMBL608402 0.81 NOS1 (0.49) NOS1
Arginine SCHEMBL1487699 0.80 NOS1 (0.52) NOS1NOS3NOS2OTCDDAH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2046 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4727356-A2 SYNTHETIC ANTIFREEZE GLYCOPROTEINS WITH ICE-BINDING ACTIVITY University of Utah Research Foundation (US) 2026-04-22 EP claimed
US-12590123-B2 Compounds and methods for treating cancer, viral infections, and allergic conditions WASHINGTON UNIVERSITY (US) 2026-03-31 US claimed
EP-4709378-A1 COMPOUNDS FOR NOS-RELATED CANCERS AND METHODS OF USE Yissum Research Development Company of the Hebrew University of Jerusalem Ltd. (IL) 2026-03-18 EP claimed
US-12520839-B2 Methods and compositions for cryopreservation of cell therapies THE GEORGE WASHINGTON UNIVERSITY (US) 2026-01-13 US claimed
EP-4649136-A1 GENETIC MODIFICATION OF MICROBES FOR PRODUCTION OF NITROGEN AND CARBON-CONTAINING COMPOUNDS Fertis India Pvt Ltd (IN) 2025-11-19 EP claimed
US-20250257093-A1 BETULASTATIN COMPOUNDS ARIZONA BOARD OF REGENTS ON BEHALF OF ARIZONA STATE UNIVERSITY 2025-08-14 US claimed
WO-2025111482-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS AT LOW STOICHIOMETRIC RATIOS BEXSON BIOMEDICAL, INC. (US) 2025-05-30 WO claimed
US-20250171495-A1 MUTLI-TARGETED SERINE PROTEASE INHIBITORS FOR TREATMENT OF CANCER AND VIRAL INFECTION WASHINGTON UNIVERSITY 2025-05-29 US claimed
EP-4554947-A1 PROTEASE/ENZYME CLEAVABLE LINKER-PAYLOADS AND PROTEIN CONJUGATES Sutro Biopharma, Inc. (US) 2025-05-21 EP claimed
CN-119948030-A Protease/enzyme cleavable linker-payload and protein conjugates 苏特罗生物制药公司 2025-05-06 CN claimed
WO-1996002241-A1 USE OF NITROGEN OXIDE SPECIES AND ADDUCTS TO INHIBIT SKELETAL MUSCLE CONTRACTION DUKE UNIVERSITY (US) 1996-02-01 WO claimed
US-5439938-A Treating priapism by applying to erect penis an inhibitor of NO synthetase to cause penis to become flaccid THE JOHNS HOPKINS UNIVERSITY (US) 1995-08-08 US claimed
EP-0603335-A4 ATTENUATION OF THE OPIOID WITHDRAWAL SYNDROME BY INHIBITORS OF NITRIC OXIDE SYNTHASE. US HEALTH (US) 1995-07-05 EP claimed
EP-0603335-A1 ATTENUATION OF THE OPIOID WITHDRAWAL SYNDROME BY INHIBITORS OF NITRIC OXIDE SYNTHASE THE GOVERNMENT OF THE UNITED STATES OF AMERICA as represented by the SECRETARY OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1994-06-29 EP claimed
US-5266594-A For treatment of stroke or nervous system disorders such as Alzheimer's disease and Huntington's disease NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 1993-11-30 US claimed
US-5212287-A Multistage synthesis of oligopeptides with protection of side groups then deprotection after reaction IMMUNETECH PHARMACEUTICALS, INC. (US) 1993-05-18 US claimed
WO-1993005775-A1 ATTENUATION OF THE OPIOID WITHDRAWAL SYNDROME BY INHIBITORS OF NITRIC OXIDE SYNTHASE THE GOVERNMENT OF THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1993-04-01 WO claimed
EP-0399885-A1 Tripeptide, its process of preparation and its use RHONE-POULENC CHIMIE (FR) 1990-11-28 EP claimed
US-4960881-A REACTING AMINO ACID WITH ALPHA-CHLORINATED CARBONATE IN SOLVENT IN PRESENCE OF ACID SCAVENGER SOCIETE NATIONALE DES POUDRES ET EXPLOSIFS (FR) 1990-10-02 US claimed
EP-0154581-B1 ALPHA-CHLORINATED CARBONATES, PROCESS FOR THEIR PREPARATION AND THEIR APPLICATION TO THE PROTECTION OF AMINIC FUNCTIONS IN AMINO ACIDS SOCIETE NATIONALE DES POUDRES ET EXPLOSIFS (FR) 1988-06-08 EP claimed