SCHEMBL3454173

SCHEMBL3454173

NC(=O)c1ccc2c(O)c(C(N)=O)ccc2c1

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LCK P06239 4/20 0.55
ERN1 O75460 2/20 0.43
PLAU P00749 3/20 0.41
PTPN11 Q06124 1/20 0.41
LDHA P00338 1/20 0.41
PARP1 P09874 1/20 0.40
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.40
GAA P10253 1/20 0.40
PTPN1 P18031 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
CSNK2A1 P68400 1/20 0.38
HIPK2 Q9H2X6 1/20 0.38
NOS1 P29475 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3028424 0.81 LCK (0.49) LCKERN1PLAUPARP1ALDH1A1
SCHEMBL19873094 0.78 ERN1 (0.57) LCKERN1PLAUALDH1A1KDM4E
SCHEMBL3454172 0.77 LCK (0.45) LCKERN1PLAUPARP1ALDH1A1
SCHEMBL29463701 0.76 ALDH1A1 (0.62) LCKPLAUPARP1ALDH1A1KDM4E
SCHEMBL3237472 0.76 PTPN1 (0.61) LCKERN1PTPN11LDHAALDH1A1
SCHEMBL6384957 0.76 ALDH1A1 (0.62) LCKPLAUPARP1ALDH1A1KDM4E
SCHEMBL2363489 0.76 LCK (0.78) LCKPLAUPARP1ALDH1A1KDM4E
SCHEMBL30394609 0.76 PLAU (0.47) LCKERN1PLAUALDH1A1KDM4E
SCHEMBL356272 0.76 LDHA (0.69) LDHAKDM4EMAPT
SCHEMBL28013895 0.74 LCK (0.42) LCKERN1PLAUPARP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2205070-A1 N-HYDROXY-NAPHTHALENE DICARBOXAMIDE AND N-HYDROXY-BIPHENYL-DICARBOXAMIDE COMPOUNDS AS HISTONE DEACETYLASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2010-07-14 EP claimed
WO-2009045385-A1 N-HYDROXY-NAPHTHALENE DICARBOXAMIDE AND N-HYDROXY-BIPHENYL-DICARBOXAMIDE COMPOUNDS AS HISTONE DEACETYLASE INHIBITORS MERCK & CO., INC. (US) 2009-04-09 WO claimed
EP-2205070-A1 N-HYDROXY-NAPHTHALENE DICARBOXAMIDE AND N-HYDROXY-BIPHENYL-DICARBOXAMIDE COMPOUNDS AS HISTONE DEACETYLASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2010-07-14 EP disclosed
WO-2009045385-A1 N-HYDROXY-NAPHTHALENE DICARBOXAMIDE AND N-HYDROXY-BIPHENYL-DICARBOXAMIDE COMPOUNDS AS HISTONE DEACETYLASE INHIBITORS MERCK & CO., INC. (US) 2009-04-09 WO disclosed