SCHEMBL3454172

SCHEMBL3454172

CC(C)c1c(C(N)=O)ccc2cc(C(N)=O)ccc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LCK P06239 2/20 0.45
ALDH1A1 P00352 3/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
PLAU P00749 3/20 0.38
ACE2 Q9BYF1 1/20 0.38
KDM4E B2RXH2 2/20 0.37
BRD4 O60885 1/20 0.37
BRPF1 P55201 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
HSD17B10 Q99714 1/20 0.37
CYP17A1 P05093 1/20 0.37
CYP3A4 P08684 1/20 0.37
ERN1 O75460 2/20 0.37
PARP10 Q53GL7 1/20 0.37
GAA P10253 1/20 0.36
CSNK2A1 P68400 1/20 0.35
HIPK2 Q9H2X6 1/20 0.35
PARP1 P09874 1/20 0.35
PTPN1 P18031 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3028424 0.79 LCK (0.49) LCKALDH1A1MAPTHPGDPLAU
SCHEMBL7477120 0.79 NCEH1 (0.54) ALDH1A1HPGDKDM4ESMN1; SMN2PARP10
SCHEMBL3454173 0.77 LCK (0.55) LCKALDH1A1MAPTHPGDPLAU
SCHEMBL2882576 0.75 IRAK4 (0.44) ALDH1A1MAPTHPGDKDM4EHSD17B10
SCHEMBL21871911 0.74 LCK (0.43) LCKMAPTPLAUCYP17A1CYP3A4
SCHEMBL19873094 0.73 ERN1 (0.57) LCKALDH1A1MAPTHPGDPLAU
SCHEMBL4405181 0.73 LCK (0.75) LCKALDH1A1MAPTPLAUKDM4E
SCHEMBL30935786 0.73 LCK (0.75) LCKALDH1A1MAPTPLAUKDM4E
SCHEMBL2976652 0.73 ACE2 (0.44) LCKALDH1A1ACE2KDM4EBRD4
SCHEMBL6384957 0.71 ALDH1A1 (0.62) LCKALDH1A1MAPTHPGDPLAU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2205070-A1 N-HYDROXY-NAPHTHALENE DICARBOXAMIDE AND N-HYDROXY-BIPHENYL-DICARBOXAMIDE COMPOUNDS AS HISTONE DEACETYLASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2010-07-14 EP claimed
WO-2009045385-A1 N-HYDROXY-NAPHTHALENE DICARBOXAMIDE AND N-HYDROXY-BIPHENYL-DICARBOXAMIDE COMPOUNDS AS HISTONE DEACETYLASE INHIBITORS MERCK & CO., INC. (US) 2009-04-09 WO claimed