SCHEMBL345469

SCHEMBL345469

O=NCCNC(=S)NCc1ccc(F)cc1C(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 13/20 0.44
NTRK1 P04629 1/20 0.43
EPHX2 P34913 3/20 0.42
HDAC3 O15379 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
PPARG P37231 2/20 0.42
IDO1 P14902 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7792525 0.84 P2RX7 (0.45) P2RX7NTRK1EPHX2HDAC3HDAC1
SCHEMBL5723612 0.73 P2RX7 (0.57) P2RX7NTRK1EPHX2HDAC3HDAC1
SCHEMBL16538118 0.70 P2RX7 (0.57) P2RX7NTRK1EPHX2HDAC3HDAC1
SCHEMBL4576232 0.70 P2RX7 (0.55) P2RX7NTRK1EPHX2HDAC3HDAC1
SCHEMBL16972742 0.70 HDAC3 (0.55) P2RX7NTRK1EPHX2HDAC3HDAC1
SCHEMBL6355300 0.69 EPHX2 (0.55) P2RX7NTRK1EPHX2HDAC3HDAC1
SCHEMBL16538163 0.68 IDO1 (0.49) P2RX7NTRK1EPHX2HDAC3HDAC1
SCHEMBL343998 0.68 LMNA (0.43)
SCHEMBL6355022 0.68 EPHX2 (0.53) P2RX7NTRK1EPHX2HDAC3HDAC1
SCHEMBL28438485 0.67 EPHX2 (0.52) EPHX2PPARGIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2428207-A1 Alpha-2B adrenergic receptor agonist and serotonin-norepinephrine reuptake inhibitor compositions for treating chronic pain Allergan, Inc. (US) 2012-03-14 EP disclosed