SCHEMBL3456724

SCHEMBL3456724

O=Cc1cc2c(=O)n(CCc3ccccc3)c(=O)n(Cc3ccc(-c4ccccc4)cc3)c2s1

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PDE1B Q01064 1/20 0.49
HDAC1 Q13547 5/20 0.48
HDAC6 Q9UBN7 5/20 0.48
HDAC11 Q96DB2 4/20 0.48
HDAC8 Q9BY41 4/20 0.48
TP53 P04637 2/20 0.48
MAPT P10636 2/20 0.48
AGTR1 P30556 4/20 0.47
MELK Q14680 1/20 0.45
LMNA P02545 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3456723 0.93 MAPT (0.50) PDE1BHDAC1HDAC6HDAC11HDAC8
SCHEMBL2774113 0.87 AGTR1 (0.48) HDAC1HDAC6HDAC11HDAC8TP53
SCHEMBL13070234 0.84 AGTR1 (0.54) PDE1BHDAC1HDAC6HDAC11HDAC8
SCHEMBL2776910 0.73 AGTR1 (0.54) PDE1BHDAC1HDAC6HDAC11HDAC8
SCHEMBL17483612 0.72 PDE1B (0.76) PDE1B
SCHEMBL2774771 0.71 AGTR1 (0.54) AGTR1
SCHEMBL18808388 0.70 PDE1B (0.52) PDE1B
SCHEMBL24031181 0.69 THRB (0.71) HDAC1HDAC6HDAC11HDAC8TP53
SCHEMBL2773612 0.69 AGTR1 (0.73) AGTR1
SCHEMBL2774054 0.68 HDAC1 (0.60) PDE1BHDAC1HDAC6HDAC11HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2253630-A1 Heterocyclic compound and use thereof Takeda Pharmaceutical Company Limited (JP) 2010-11-24 EP disclosed