SCHEMBL3456723

SCHEMBL3456723

O=Cc1cc2c(=O)n(CCc3ccccc3)c(=O)n(Cc3cccc(-c4ccccc4)c3)c2s1

nearest known ligand 0.50

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.50
TP53 P04637 3/20 0.50
HDAC8 Q9BY41 3/20 0.45
HDAC6 Q9UBN7 3/20 0.45
HDAC1 Q13547 1/20 0.43
HDAC11 Q96DB2 1/20 0.43
CASR P41180 2/20 0.42
PDE1B Q01064 1/20 0.42
ADORA2B P29275 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3456724 0.93 PDE1B (0.49) MAPTTP53HDAC8HDAC6HDAC1
SCHEMBL2774113 0.80 AGTR1 (0.48) MAPTTP53HDAC8HDAC6HDAC1
SCHEMBL13070234 0.77 AGTR1 (0.54) MAPTTP53HDAC8HDAC6HDAC1
SCHEMBL17483612 0.69 PDE1B (0.76) PDE1B
SCHEMBL18808388 0.68 PDE1B (0.52) PDE1B
SCHEMBL16637309 0.67 HTT (0.52) MAPTTP53HDAC8HDAC6HDAC1
SCHEMBL2776910 0.66 AGTR1 (0.54) HDAC8HDAC6HDAC1HDAC11PDE1B
SCHEMBL19611087 0.64 ADORA2B (0.53) HDAC8HDAC6HDAC1HDAC11ADORA2B
SCHEMBL24031181 0.64 THRB (0.71) MAPTTP53HDAC8HDAC6HDAC1
SCHEMBL16643997 0.64 ADORA2B (0.56) MAPTTP53HDAC8HDAC6HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2253630-A1 Heterocyclic compound and use thereof Takeda Pharmaceutical Company Limited (JP) 2010-11-24 EP disclosed