Cholrphenethazine

Cholrphenethazine

SCHEMBL3456873

CN(C)CCN1c2ccccc2Sc2ccc(Cl)cc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 1/20 1.00
ICAM1 P05362 1/20 1.00
ITGAL P20701 1/20 1.00
CYP1A2 P05177 7/20 0.85
CYP2D6 P10635 7/20 0.85
CYP2C19 P33261 5/20 0.85
HTR1A P08908 5/20 0.85
DRD2 P14416 4/20 0.85
LMNA P02545 4/20 0.85
MAPT P10636 4/20 0.85
SMN1; SMN2 Q16637 4/20 0.85
TP53 P04637 4/20 0.85
CHRM2 P08172 4/20 0.85
ADRA2A P08913 4/20 0.85
CHRM1 P11229 4/20 0.85
DRD1 P21728 4/20 0.85
SLC6A2 P23975 4/20 0.85
SLC6A4 P31645 4/20 0.85
ADRA1A P35348 4/20 0.85
OPRM1 P35372 4/20 0.85

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cholrphenethazine SCHEMBL29376339 0.99 ITGB2 (0.97) ITGB2ICAM1ITGALCYP1A2CYP2D6
Cholrphenethazine SCHEMBL9724481 0.99 ITGB2 (0.97) ITGB2ICAM1ITGALCYP1A2CYP2D6
Chlorpromazine SCHEMBL29358018 0.92 CYP1A2 (1.00) ITGB2ICAM1ITGALCYP1A2CYP2D6
Chlorpromazine SCHEMBL29367385 0.92 CYP1A2 (1.00) ITGB2ICAM1ITGALCYP1A2CYP2D6
Chlorpromazine SCHEMBL8321 0.92 CYP1A2 (1.00) ITGB2ICAM1ITGALCYP1A2CYP2D6
Chlorpromazine SCHEMBL23326209 0.91 CYP1A2 (1.00) ITGB2ICAM1ITGALCYP1A2CYP2D6
Chlorpromazine SCHEMBL5483904 0.91 CYP1A2 (1.00) ITGB2ICAM1ITGALCYP1A2CYP2D6
Chlorpromazine SCHEMBL41771 0.91 CYP1A2 (1.00) ITGB2ICAM1ITGALCYP1A2CYP2D6
SCHEMBL9724480 0.91 CYP1A2 (0.93) ITGB2ICAM1ITGALCYP1A2CYP2D6
Chlorpromazine SCHEMBL29351728 0.91 CYP1A2 (1.00) ITGB2ICAM1ITGALCYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1976723-A Treatment of infectious diseases BKG PHARMA APS (DK) 2007-06-06 CN claimed
EP-1744781-A1 TREATMENT OF INFECTIOUS DISEASES Bkg Pharma Aps (DK) 2007-01-24 EP claimed
WO-2005105145-A1 TREATMENT OF INFECTIOUS DISEASES BKG PHARMA APS (DK) 2005-11-10 WO claimed
EP-1744781-B1 TREATMENT OF INFECTIOUS DISEASES BKG PHARMA APS (DK) 2012-07-04 EP disclosed
CN-1976723-B Use of preparing medicine for treating or preventing infectious diseases BKG PHARMA APS 2010-12-29 CN disclosed
EP-2260870-A2 Treatment of infectious diseases with combinations of a thioxanthene derivative with an anti-infective agent BKG Pharma ApS (DK) 2010-12-15 EP disclosed
US-20080318970-A1 Treatment of Infectious Diseases BKG PHARMA APS (DK) 2008-12-25 US disclosed
CN-1976723-A Treatment of infectious diseases BKG PHARMA APS (DK) 2007-06-06 CN disclosed
EP-1744781-A1 TREATMENT OF INFECTIOUS DISEASES Bkg Pharma Aps (DK) 2007-01-24 EP disclosed
WO-2005105145-A1 TREATMENT OF INFECTIOUS DISEASES BKG PHARMA APS (DK) 2005-11-10 WO disclosed
US-5104858-A Administering trans-flupenthiyol with doxorubicin; lack of antipsychotic activity reduces side effects YALE UNIVERSITY (US) 1992-04-14 US disclosed
EP-0361485-A2 A method of sensitizing multidrug resistant cells to antitumor agents YALE UNIVERSITY (US) 1990-04-04 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080318970-A1 Treatment of Infectious Diseases ABCC1, TST, TPMT ITGB2 4165/4885ICAM1 931/4885ITGAL 3376/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.