SCHEMBL3459072

SCHEMBL3459072

[O]c1cc(C(F)(F)F)ccc1F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.44
PDE2A O00408 3/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
CES2 O00748 3/20 0.41
TSHR P16473 1/20 0.40
MPL P40238 1/20 0.40
PTPN5 P54829 1/20 0.39
NOS3 P29474 1/20 0.39
NOS2 P35228 1/20 0.39
EPHX2 P34913 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
HSD17B10 Q99714 1/20 0.38
TMPRSS4 Q9NRS4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2839879 0.81 PDE2A (0.47) IDO1PDE2AMEN1KMT2ACES2
SCHEMBL29827588 0.77 PDE2A (0.50) IDO1PDE2AMEN1KMT2ACES2
SCHEMBL2147584 0.77 PDE2A (0.50) IDO1PDE2AMEN1KMT2ACES2
SCHEMBL30568357 0.75 MPL (0.55) IDO1PDE2ACES2TSHRMPL
SCHEMBL18361131 0.75 MPL (0.55) IDO1PDE2ACES2TSHRMPL
SCHEMBL2459420 0.75 PDE2A (0.48) IDO1PDE2AMEN1KMT2ACES2
SCHEMBL3760427 0.74 ALDH1A1 (0.45) PDE2AMEN1KMT2ACES2TSHR
SCHEMBL476625 0.73 PDE2A (0.47) IDO1PDE2AMPLPTPN5TRPA1
SCHEMBL2699647 0.73 CES2 (0.52) IDO1PDE2AMEN1KMT2ACES2
SCHEMBL30417923 0.73 CES2 (0.52) IDO1PDE2AMEN1KMT2ACES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8426631-B2 Fungicidal compounds, method for the production thereof, and use thereof to combat damaging fungi, and agents comprising the same BASF SE (DE) 2013-04-23 US disclosed
EP-2264010-A1 Hetarylamidines Bayer CropScience AG (DE) 2010-12-22 EP disclosed
US-20100304966-A1 Fungicidal Compounds, Method For the Production Thereof, And Use Thereof To Combat Damaging Fungi, And Agents Comprising The Same BASF SE (DE) 2010-12-02 US disclosed
US-7592352-B2 Substituted thieno and furo-pyridines SMITHKLINE BEECHAM CORPORATION (US) 2009-09-22 US disclosed
US-20080182868-A1 Novel chemical compounds SMITHKLINE BEECHAM CORPORATION 2008-07-31 US disclosed
EP-1620094-A2 NOVEL CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-02-01 EP disclosed
WO-2004100947-A2 NOVEL CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2004-11-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080182868-A1 Novel chemical compounds HRAS, VHL, TP53 IDO1 4024/4885PDE2A 3748/4885MEN1 1739/4885
US-20100304966-A1 Fungicidal Compounds, Method For the Production Thereof, And Use Thereof To Combat Damaging Fungi, And Agents Comprising The Same CYP51A1, ERG28, CAT IDO1 753/4885PDE2A 223/4885MEN1 1227/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.