SCHEMBL3462

SCHEMBL3462

CN(C)CCc1sccc1CO

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.42
HTR2C P28335 3/20 0.42
HTR2B P41595 3/20 0.42
HRH1 P35367 1/20 0.37
TAAR1 Q96RJ0 6/20 0.35
HRH3 Q9Y5N1 1/20 0.35
LTB4R Q15722 6/20 0.35
HTR1A P08908 1/20 0.34
HTR6 P50406 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4743163 0.85 HTR2A (0.46) HTR2AHTR2CHTR2BTAAR1HRH3
SCHEMBL5109988 0.79 LTB4R (0.34) LTB4R
SCHEMBL5104355 0.78 LTB4R (0.36) LTB4R
SCHEMBL2085294 0.78 LTB4R (0.41) HTR2CLTB4R
SCHEMBL27277657 0.77 HTR2A (0.41) HTR2AHTR2CHTR2BHRH1TAAR1
SCHEMBL2690986 0.75
SCHEMBL6050537 0.75 KDM4E (0.34) LTB4R
SCHEMBL5104136 0.74
SCHEMBL5799093 0.73 ALDH1A1 (0.39) HRH3
SCHEMBL27720648 0.73 HTR2A (0.41) HTR2AHTR2CHTR2BHRH1TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5023269-A 3-aryloxy-3-substituted propanamines ELI LILLY AND COMPANY (US) 1991-06-11 US disclosed
EP-0273658-B1 3-ARYLOXY-3-SUBSTITUTED PROPANAMINES ELI LILLY AND COMPANY (US) 1990-10-31 EP disclosed
US-4956388-A ANTIDEPRESSANTS, ANTIANXIETY, TREATMENT OF OBESITY, ADDICTION TO SMOKING AND ALCOHOL ELI LILLY AND COMPANY (US) 1990-09-11 US disclosed
EP-0273658-A1 3-Aryloxy-3-substituted propanamines ELI LILLY AND COMPANY (US) 1988-07-06 EP disclosed