SCHEMBL3465091

SCHEMBL3465091

CN(C)CCNc1ccc(C(N)=O)cn1

nearest known ligand 0.62

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NNMT P40261 1/20 0.58
HCAR3 P49019 5/20 0.52
RET P07949 1/20 0.52
EPHX2 P34913 1/20 0.51
CYP2C19 P33261 1/20 0.49
HRH3 Q9Y5N1 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5140766 0.84 HCAR3 (0.55) HCAR3CYP2C19HRH3
SCHEMBL30737636 0.84 HCAR3 (0.55) HCAR3CYP2C19HRH3
SCHEMBL5205802 0.81 NNMT (0.60) NNMTHCAR3EPHX2
SCHEMBL30492154 0.80 NNMT (0.58) NNMTHCAR3EPHX2
SCHEMBL11546416 0.80 HCAR3 (0.73) NNMTHCAR3EPHX2
SCHEMBL12953967 0.79 HCAR3 (0.76) NNMTHCAR3EPHX2
SCHEMBL1680894 0.79 HCAR3 (0.76) NNMTHCAR3EPHX2
SCHEMBL1937770 0.78 HCAR3 (0.57) NNMTHCAR3EPHX2
SCHEMBL3464039 0.77 NNMT (0.55) NNMTHCAR3EPHX2
SCHEMBL29036800 0.76 CYP2C19 (0.56) HCAR3CYP2C19HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346868-B1 AZAINDAZOLE COMPOUNDS AS CCR1 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2016-01-27 EP disclosed
US-8338610-B2 Pyridinyl compounds useful as intermediates BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-12-25 US disclosed
US-20120136158-A1 Pyridinyl Compounds Useful As Intermediates BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-05-31 US disclosed
US-20100093724-A1 Azaindazole Compounds As CCR1 Receptor Antagonists BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-04-15 US disclosed
US-4203988-A ANTISECRETORY AGENTS MERCK & CO., INC. (US) 1980-05-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100093724-A1 Azaindazole Compounds As CCR1 Receptor Antagonists CCR1, CCR3, CCR4 NNMT 1562/4885HCAR3 46/4885RET 2995/4885
US-20120136158-A1 Pyridinyl Compounds Useful As Intermediates CCR1, CCRL2, CCR4 NNMT 957/4885HCAR3 450/4885RET 4351/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.