Methylprednisolone Aceponate

Methylprednisolone Aceponate

SCHEMBL3466

CCC(=O)O[C@]1(C(=O)COC(C)=O)CC[C@H]2[C@@H]3C[C@H](C)C4=CC(=O)C=C[C@]4(C)[C@H]3[C@@H](O)C[C@@]21C

nearest known ligand 0.74

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 8/20 0.74
CYP3A4 P08684 5/20 0.74
AR P10275 2/20 0.74
F2 P00734 1/20 0.74
NR3C1 P04150 7/20 0.63
HIF1A Q16665 7/20 0.60
ABCB11 O95342 3/20 0.60
NR1I2 O75469 2/20 0.60
ALDH1A1 P00352 2/20 0.60
HSD17B10 Q99714 1/20 0.60
ABCC4 O15439 1/20 0.60
PDE4D Q08499 1/20 0.60
CHRM1 P11229 1/20 0.60
LMNA P02545 4/20 0.60
USP2 O75604 3/20 0.60
CYP2C9 P11712 2/20 0.60
CYP2D6 P10635 1/20 0.60
NPSR1 Q6W5P4 1/20 0.52
NR3C2 P08235 1/20 0.48
ABCC3 O15438 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Methylprednisolone Aceponate SCHEMBL8961317 1.00 PGR (0.74) PGRCYP3A4ARF2NR3C1
Methylprednisolone Aceponate SCHEMBL8612416 1.00 PGR (0.74) PGRCYP3A4ARF2NR3C1
SCHEMBL10910516 0.95 PGR (0.67) PGRCYP3A4ARF2NR3C1
SCHEMBL10910515 0.95 PGR (0.67) PGRCYP3A4ARF2NR3C1
SCHEMBL10881968 0.94 PGR (0.72) PGRCYP3A4ARF2NR3C1
SCHEMBL10934308 0.94 PGR (0.72) PGRCYP3A4ARF2NR3C1
SCHEMBL10881975 0.94 PGR (0.72) PGRCYP3A4ARF2NR3C1
SCHEMBL10902829 0.94 PGR (0.69) PGRCYP3A4ARF2NR3C1
SCHEMBL10902825 0.94 PGR (0.69) PGRCYP3A4ARF2NR3C1
SCHEMBL10906704 0.94 PGR (0.79) PGRCYP3A4ARF2NR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3232 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4710918-A1 OPHTHALMIC PHARMACEUTICAL COMPOSITION AND PREPARATION METHOD THEREFOR, OPHTHALMIC KIT CONTAINING OPHTHALMIC PHARMACEUTICAL COMPOSITION, AND USE Shenyang Xingqi Pharmaceutical Co., Ltd. (CN) 2026-03-18 EP claimed
US-20250255781-A1 PROCESSES FOR PREPARATION OF 3-D PRINTED PHARMACEUTICAL PRODUCTS BRISTOL-MYERS SQUIBB COMPANY (US) 2025-08-14 US claimed
US-12296043-B2 Liquisoft capsules PATHEON SOFTGELS INC. (US) 2025-05-13 US claimed
WO-2025090570-A1 ANTI-OX40L ANTIBODIES AND METHODS OF USE ABCELLERA BIOLOGICS INC. (CA) 2025-05-01 WO claimed
EP-4510999-A1 PROCESSES FOR PREPARATION OF 3-D PRINTED PHARMACEUTICAL PRODUCTS Bristol-Myers Squibb Company (US) 2025-02-26 EP claimed
US-20250032513-A1 Ophthalmic Pharmaceutical Composition, Ophthalmic Kit, and Pharmaceutical Application Thereof SHENYANG XINGQI PHARMACEUTICAL CO., LTD. (CN) 2025-01-30 US claimed
CN-119212681-A Method for preparing 3-D printed pharmaceutical products 百时美施贵宝公司 2024-12-27 CN claimed
CN-118955596-A Methylprednisolone aceponate preparation method of nylon 河南利华制药有限公司 2024-11-15 CN claimed
US-20240360210-A1 USE OF AN IL-18 ANTAGONIST FOR TREATING AND/OR PREVENTION OF ATOPIC DERMATITIS OR A RELATED CONDITION NOVARTIS PHARMA AG (CH) 2024-10-31 US claimed
EP-4426355-A1 GLYCOSYLATED PRODRUGS Universiteit Leiden (NL) 2024-09-11 EP claimed
CN-1179721-A Novel pharmaceutical formulations ASTRA AB (SE) 1998-04-22 CN claimed
CN-1179718-A Novel pharmaceutical composition ASTRA AB (SE) 1998-04-22 CN claimed
EP-0809501-A1 NOVEL PHARMACEUTICAL FORMULATION Astra Aktiebolag (SE) 1997-12-03 EP claimed
EP-0809498-A1 NOVEL PHARMACEUTICAL COMBINATION Astra Aktiebolag (SE) 1997-12-03 EP claimed
WO-1996024359-A1 NOVEL PHARMACEUTICAL FORMULATION ASTRA AKTIEBOLAG (SE) 1996-08-15 WO claimed
WO-1996024355-A1 NOVEL PHARMACEUTICAL COMBINATION ASTRA AKTIEBOLAG (SE) 1996-08-15 WO claimed
EP-0675722-A1 HYDROXY VITAMIN D3 COMPOUNDS FOR TREATING SKIN ATROPHY LEO PHARMACEUTICAL PRODUCTS LTD. A/S (LOVENS KEMISKE FABRIK PRODUKTIONSAKTIESELSKAB) (DK) 1995-10-11 EP claimed
WO-1994014453-A1 HYDROXY VITAMIN D3 COMPOUNDS FOR TREATING SKIN ATROPHY Leo Pharmaceutical Products Ltd. A/S (Løvens Kemiske Fabrik Produktionsaktieselskab) (DK) 1994-07-07 WO claimed
EP-0072547-B1 6-ALPHA-METHYL-PREDNISOLONE DERIVATIVES, THEIR PREPARATION AND UTILIZATION SCHERING AKTIENGESELLSCHAFT (DE) 1986-03-26 EP claimed
EP-0095894-A2 6 Alpha-methylprednisolone derivatives OHTA SEIYAKU KABUSHIKI KAISHA. (JP) 1983-12-07 EP claimed