SCHEMBL3466282

SCHEMBL3466282

NC(=O)c1ccc(NC(=O)C2CC2)nc1

nearest known ligand 0.63

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NNMT P40261 1/20 0.58
NPC1 O15118 3/20 0.55
RAB9A P51151 3/20 0.55
ALDH1A1 P00352 2/20 0.55
ABL1 P00519 1/20 0.52
DEGS1 O15121 2/20 0.51
EPHX2 P34913 1/20 0.51
MAPT P10636 1/20 0.50
TP53 P04637 1/20 0.50
PKM P14618 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30498440 0.85 HCAR3 (0.66) NPC1RAB9AALDH1A1DEGS1
SCHEMBL21061901 0.85 HCAR3 (0.66) NPC1RAB9AALDH1A1DEGS1
SCHEMBL18839009 0.85 NPC1 (0.50) NPC1RAB9AALDH1A1DEGS1MAPT
SCHEMBL18839006 0.85 NPC1 (0.50) NPC1RAB9AALDH1A1DEGS1MAPT
SCHEMBL30636222 0.81 NNMT (0.51) NNMTALDH1A1EPHX2
SCHEMBL29686685 0.81 KMT2A (0.54) NPC1RAB9AALDH1A1ABL1DEGS1
SCHEMBL25702959 0.80 NPC1 (0.51) NPC1RAB9AALDH1A1ABL1DEGS1
SCHEMBL28847350 0.80 NPC1 (0.54) NPC1RAB9AALDH1A1ABL1DEGS1
SCHEMBL29874618 0.80 NPC1 (0.54) NPC1RAB9AALDH1A1ABL1DEGS1
SCHEMBL5239807 0.79 HCAR3 (0.68) NPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112047928-B Isonicotinamide AChE-GSK3 double inhibitor and preparation method and application thereof 中国药科大学 2022-09-23 CN disclosed
WO-2022105771-A1 NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVE, AND PREPARATION METHOD THEREFOR AND MEDICAL APPLICATION THEREOF 江苏恒瑞医药股份有限公司 2022-05-27 WO disclosed
CN-112047928-A Isonicotinamide AChE-GSK3 double inhibitor and preparation method and application thereof 中国药科大学 2020-12-08 CN disclosed
EP-2346868-B1 AZAINDAZOLE COMPOUNDS AS CCR1 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2016-01-27 EP disclosed
US-20100093724-A1 Azaindazole Compounds As CCR1 Receptor Antagonists BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-04-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100093724-A1 Azaindazole Compounds As CCR1 Receptor Antagonists CCR1, CCR3, CCR4 NNMT 1562/4885NPC1 2064/4885RAB9A 2908/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.