SCHEMBL3466941

SCHEMBL3466941

CC(C)C[C@@H](C#N)OS(=O)(=O)c1ccc(Br)cc1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSK P43235 6/20 0.40
MMP1 P03956 1/20 0.39
MMP2 P08253 1/20 0.39
MMP3 P08254 1/20 0.39
MMP7 P09237 1/20 0.39
MMP9 P14780 1/20 0.39
MMP13 P45452 1/20 0.39
PLCG1 P19174 1/20 0.36
CTSB P07858 3/20 0.33
CA2 P00918 1/20 0.33
FPR2 P25090 1/20 0.33
CYP1A1 P04798 1/20 0.33
CTSL P07711 2/20 0.33
CTSS P25774 2/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3466693 0.87 CA1 (0.40) CA2ALDH1A1
SCHEMBL3467086 0.85 MEN1 (0.39) CTSKCTSBCA2CTSLCTSS
SCHEMBL3466268 0.85 CTSL (0.40) CTSKCTSBCTSLCTSSALDH1A1
SCHEMBL27821616 0.85 CTSL (0.40) CTSKCTSBCTSLCTSSALDH1A1
SCHEMBL3466972 0.82 CA9 (0.39) MMP1MMP2MMP9MMP13CA2
SCHEMBL3466897 0.74 KMT2A (0.47) MMP1MMP2MMP9MMP13CA2
SCHEMBL18853809 0.73 CA2 (0.45) MMP1MMP2MMP3MMP7MMP9
SCHEMBL13296183 0.71 PLCG1 (0.42) MMP1MMP2MMP3MMP7MMP9
SCHEMBL7694180 0.71 PLCG1 (0.42) MMP1MMP2MMP3MMP7MMP9
SCHEMBL28928743 0.71 GLA (0.41) CA2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010070593-A2 MALONATE ESTERS PFIZER IRELAND PHARMACEUTICALS (IE) 2010-06-24 WO disclosed
WO-2010070593-A2 MALONATE ESTERS PFIZER IRELAND PHARMACEUTICALS (IE) 2010-06-24 WO disclosed