SCHEMBL3467798

SCHEMBL3467798

Nc1cc(CC=O)c(Cl)cc1Br

nearest known ligand 0.31

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA9 Q16790 1/20 0.31
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21052503 0.78 AHR (0.36) CA1CA2CA9GAA
SCHEMBL26601688 0.78
SCHEMBL21356184 0.76 AHR (0.32)
SCHEMBL29384228 0.76 AHR (0.32)
SCHEMBL3344291 0.75 GAA (0.33) CA1CA2CA9GAA
SCHEMBL27749404 0.73 ALDH1A1 (0.32)
SCHEMBL4591472 0.72 GAA (0.40) CA1CA2CA9GAA
SCHEMBL3468380 0.72 MEN1 (0.34) GAA
SCHEMBL29951151 0.71 TDP1 (0.42) CA1CA2CA9GAA
SCHEMBL3467784 0.71 CYP3A4 (0.48) CA1CA2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2393781-A1 DIHYDROPYRIDONE UREAS AS P2X7 MODULATORS F. Hoffmann-La Roche AG (CH) 2011-12-14 EP disclosed
WO-2010072599-A1 DIHYDROPYRIDONE UREAS AS P2X7 MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2010-07-01 WO disclosed