SCHEMBL4591472

SCHEMBL4591472

Nc1cc(Cl)c(Cl)cc1CC=O

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.40
CD44 P16070 1/20 0.33
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA3 P07451 1/20 0.32
CA4 P22748 1/20 0.32
CA6 P23280 1/20 0.32
CA5A P35218 1/20 0.32
CA7 P43166 1/20 0.32
CA9 Q16790 1/20 0.32
CA14 Q9ULX7 1/20 0.32
CA5B Q9Y2D0 1/20 0.32
SIGMAR1 Q99720 1/20 0.31
ALDH1A1 P00352 1/20 0.31
CYP3A4 P08684 2/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21052503 0.84 AHR (0.36) GAACA1CA2CA9
SCHEMBL27749404 0.84 ALDH1A1 (0.32) ALDH1A1
SCHEMBL577652 0.80 GAA (0.55) GAAALDH1A1
SCHEMBL21546534 0.78 GAA (0.40) GAACD44CYP3A4TSHR
SCHEMBL588062 0.77 CYP3A4 (0.48) GAAALDH1A1CYP3A4TSHR
SCHEMBL4647358 0.75 CYP3A4 (0.46) ALDH1A1CYP3A4TSHR
SCHEMBL12963082 0.75 GAA (0.46) GAACD44CA12CA1CA2
SCHEMBL29384228 0.74 AHR (0.32) ALDH1A1
SCHEMBL8460064 0.74 IMPDH2 (0.33) ALDH1A1
SCHEMBL21356184 0.74 AHR (0.32) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1871748-A1 (3,4-DIHYDRO-QUINAZOLIN-2-YL)-INDAN-1-YL-AMINES F. Hoffmann-Roche AG (CH) 2008-01-02 EP disclosed
WO-2006108773-A1 (3,4-DIHYDRO-QUINAZOLIN-2-YL)-INDAN-1-YL-AMINES F. HOFFMANN-LA ROCHE AG (CH) 2006-10-19 WO disclosed