SCHEMBL3468129

SCHEMBL3468129

O=C1CCc2cc(-c3cccc(OC(F)(F)F)c3)ccc2N1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 5/20 0.69
CYP11B1 P15538 4/20 0.54
CYP11B2 P19099 4/20 0.54
CYP1A2 P05177 2/20 0.54
CYP2C9 P11712 2/20 0.54
TBXAS1 P24557 1/20 0.54
PDE3B Q13370 1/20 0.54
PDE3A Q14432 1/20 0.54
OTUD7B Q6GQQ9 2/20 0.53
GRIA1 P42261 1/20 0.49
CACNG8 Q8WXS5 1/20 0.49
HRH3 Q9Y5N1 1/20 0.47
MAPT P10636 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
PGR P06401 1/20 0.45
MAOA P21397 3/20 0.44
MAOB P27338 3/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2B6 P20813 1/20 0.44
CYP2C19 P33261 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3310995 0.88 KIF11 (0.70) KIF11CYP11B1CYP11B2CYP1A2CYP2C9
SCHEMBL30122307 0.85 KIF11 (0.73) KIF11MAPTSMN1; SMN2MAOAMAOB
SCHEMBL28956489 0.85 KIF11 (0.73) KIF11MAPTSMN1; SMN2MAOAMAOB
SCHEMBL24314993 0.83 CYP1A2 (0.70) KIF11CYP11B1CYP11B2CYP1A2CYP2C9
SCHEMBL16208447 0.81 KIF11 (1.00) KIF11MAPTSMN1; SMN2
SCHEMBL3315694 0.80 KIF11 (0.79) KIF11CYP11B1CYP11B2CYP1A2CYP2C9
SCHEMBL3466905 0.80 OTUD7B (0.52) KIF11CYP11B1CYP11B2OTUD7BGRIA1
SCHEMBL24314020 0.79 CYP11B1 (0.55) KIF11CYP11B1CYP11B2CYP1A2CYP2C9
SCHEMBL3309677 0.78 KIF11 (0.62) KIF11CYP11B1CYP11B2CYP1A2CYP2C9
SCHEMBL6968452 0.77 HRH3 (0.57) CYP11B1CYP11B2CYP1A2OTUD7BHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010074807-A1 3, 4-DIHYDROQUINOLIN-2 ( 1H ) -ONE DERIVATIVES AS SODIUM CHANNEL MODULATORS GILEAD PALO ALTO, INC. (US) 2010-07-01 WO disclosed